SCHEMBL5308335

SCHEMBL5308335

NC(=O)C(Br)c1nc2ccccc2s1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.57
HPGD P15428 4/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
HIF1A Q16665 1/20 0.51
HSD17B10 Q99714 1/20 0.51
LOXL2 Q9Y4K0 1/20 0.50
APEX1 P27695 2/20 0.48
RAB9A P51151 3/20 0.46
ALDH1A1 P00352 4/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
TSHR P16473 2/20 0.43
GAA P10253 2/20 0.43
MAPK1 P28482 1/20 0.43
ALOX15 P16050 1/20 0.43
CASP1 P29466 1/20 0.43
MAPT P10636 1/20 0.43
ADORA1 P30542 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29500244 1.00 ALOX5 (0.57) ALOX5HPGDCYP1A2CYP2C9CYP2C19
SCHEMBL11697365 0.82 HPGD (0.60) ALOX5HPGDCYP1A2CYP2C9CYP2C19
SCHEMBL29120812 0.81 ALOX5 (0.57) ALOX5HPGDCYP1A2CYP2C9CYP2C19
SCHEMBL11587666 0.81 ALOX5 (0.65) ALOX5HPGDCYP1A2CYP2C9CYP2C19
SCHEMBL8275741 0.79 HPGD (0.65) ALOX5HPGDCYP1A2CYP2C9CYP2C19
SCHEMBL29500235 0.79 RAB9A (0.50) HPGDHSD17B10APEX1RAB9AALDH1A1
SCHEMBL11585822 0.78 HPGD (0.60) ALOX5HPGDCYP1A2CYP2C9CYP2C19
SCHEMBL21802341 0.77 ALOX5 (0.57) ALOX5HPGDCYP1A2CYP2C9CYP2C19
SCHEMBL29500257 0.76 CYP1A2 (0.54) HPGDCYP1A2CYP2C19HSD17B10RAB9A
SCHEMBL11165753 0.75 ALOX5 (0.62) ALOX5HPGDCYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007045962-A2 NOVEL HDAC INHIBITORS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-04-26 WO disclosed