SCHEMBL5308356

SCHEMBL5308356

NCC(Cc1ccc(Cl)cc1)c1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.54
CHRNA4 P43681 1/20 0.54
GABBR2 O75899 7/20 0.50
GABBR1 Q9UBS5 7/20 0.50
LMNA P02545 3/20 0.50
CYP2C9 P11712 2/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
CYP1A2 P05177 2/20 0.50
THRB P10828 2/20 0.50
CYP3A4 P08684 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
NFKB1 P19838 1/20 0.50
DRD3 P35462 1/20 0.50
BLM P54132 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C19 P33261 1/20 0.50
TSHR P16473 1/20 0.50
SLC6A4 P31645 1/20 0.48
SLC6A2 P23975 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8621230 0.86 GABBR2 (0.53) GABBR2GABBR1SLC6A4SLC6A2SLC6A3
SCHEMBL8810284 0.86 GABBR2 (0.53) GABBR2GABBR1SLC6A4SLC6A2SLC6A3
SCHEMBL1541691 0.86 GABBR2 (0.53) GABBR2GABBR1SLC6A4SLC6A2SLC6A3
Hydrochloric Acid SCHEMBL1983404 0.84 GABBR2 (0.52) GABBR2GABBR1SLC6A4SLC6A2SLC6A3
SCHEMBL10513800 0.84 TAAR1 (0.47) GABBR2GABBR1SLC6A4SLC6A2SLC6A3
Hydrochloric Acid SCHEMBL9735022 0.82 TAAR1 (0.46) GABBR2GABBR1SLC6A4SLC6A2SLC6A3
Hydrochloric Acid SCHEMBL9735324 0.81 CHRNB2 (0.55) CHRNB2CHRNA4GABBR2GABBR1LMNA
SCHEMBL15903897 0.81 ESR1 (0.55) GABBR2GABBR1SLC6A2TAAR1
SCHEMBL5721773 0.81 ESR1 (0.55) CHRNB2CHRNA4LMNAMEN1KMT2A
SCHEMBL11861767 0.81 MEN1 (0.48) CHRNB2CHRNA4MEN1KMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007017652-A2 ARYLAKYLAMINES FOR THE TREATMENT OF CANCER ASTRAZENECA AB (SE) 2007-02-15 WO claimed
EP-2948135-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF PERVASIVE DEVELOPMENT DISORDERS Case Western Reserve University (US) 2015-12-02 EP disclosed
WO-2014117089-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF PERVASIVE DEVELOPMENT DISORDERS CASE WESTERN RESERVE UNIVERSITY (US) 2014-07-31 WO disclosed
WO-2007017652-A2 ARYLAKYLAMINES FOR THE TREATMENT OF CANCER ASTRAZENECA AB (SE) 2007-02-15 WO disclosed