SCHEMBL5309136

SCHEMBL5309136

CCOC(=O)c1cn(-c2ccc(-c3cc4ncccn4n3)cc2)nc1N(C(=O)c1ccc(Br)cc1F)C(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 6/20 0.40
CA9 Q16790 6/20 0.40
RAB9A P51151 4/20 0.39
NPC1 O15118 4/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
MAPT P10636 2/20 0.38
TP53 P04637 2/20 0.38
NPSR1 Q6W5P4 2/20 0.37
MAPK1 P28482 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.35
NFKB1 P19838 2/20 0.35
NFKB2 Q00653 2/20 0.35
RELA Q04206 2/20 0.35
LMNA P02545 1/20 0.35
ALDH1A1 P00352 3/20 0.34
GLA P06280 1/20 0.34
KDM4E B2RXH2 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14542210 0.94 CA12 (0.41) CA12CA9RAB9ANPC1MEN1
SCHEMBL5312718 0.92 TP53 (0.42) CA12CA9RAB9ANPC1MEN1
SCHEMBL5308815 0.91 APOBEC3A (0.33) MEN1KMT2AMAPTALDH1A1HPGD
SCHEMBL5309300 0.88 NPC1 (0.40) CA12CA9RAB9ANPC1MEN1
SCHEMBL5371592 0.87 CA12 (0.40) CA12CA9RAB9ANPC1MEN1
SCHEMBL14542427 0.86 NPC1 (0.45) CA12CA9RAB9ANPC1MEN1
SCHEMBL14542324 0.86 TP53 (0.41) CA12CA9RAB9ANPC1MEN1
SCHEMBL5370148 0.85 TP53 (0.44) CA12CA9RAB9ANPC1MEN1
SCHEMBL5309170 0.84 APOBEC3A (0.34) CA12CA9MEN1KMT2AMAPT
SCHEMBL5372491 0.84 NPSR1 (0.39) CA12CA9RAB9ANPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007039146-A1 4-CARBOXY PYRAZOLE DERIVATIVES AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2007-04-12 WO disclosed
WO-2007039146-A1 4-CARBOXY PYRAZOLE DERIVATIVES AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2007-04-12 WO disclosed