SCHEMBL5370148

SCHEMBL5370148

CCOC(=O)c1cn(-c2ccc(-c3cc4ncccn4n3)cc2)nc1N(C(=O)c1ccc(Cl)cc1)C(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.44
RXFP1 Q9HBX9 1/20 0.44
NPC1 O15118 5/20 0.42
RAB9A P51151 4/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
NPSR1 Q6W5P4 2/20 0.41
MAPK1 P28482 1/20 0.41
CA12 O43570 5/20 0.40
CA9 Q16790 5/20 0.40
KDM4E B2RXH2 3/20 0.39
CHEK1 O14757 1/20 0.39
EGFR P00533 1/20 0.39
KDR P35968 1/20 0.39
ALDH1A1 P00352 2/20 0.39
GLA P06280 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
MAPT P10636 5/20 0.38
THRB P10828 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14542427 0.94 NPC1 (0.45) TP53RXFP1NPC1RAB9ASMN1; SMN2
SCHEMBL14542324 0.92 TP53 (0.41) TP53RXFP1NPC1RAB9ASMN1; SMN2
SCHEMBL5371592 0.91 CA12 (0.40) TP53RXFP1NPC1RAB9ASMN1; SMN2
SCHEMBL5312718 0.91 TP53 (0.42) TP53RXFP1NPC1RAB9ASMN1; SMN2
SCHEMBL5372491 0.90 NPSR1 (0.39) NPC1RAB9ASMN1; SMN2NPSR1MAPK1
SCHEMBL5309593 0.90 HPGD (0.39) TP53NPC1RAB9ASMN1; SMN2CA12
SCHEMBL5309300 0.88 NPC1 (0.40) TP53RXFP1NPC1RAB9ASMN1; SMN2
SCHEMBL14542210 0.87 CA12 (0.41) TP53RXFP1NPC1RAB9ASMN1; SMN2
SCHEMBL5309402 0.86 CA12 (0.37) TP53RXFP1NPC1RAB9ASMN1; SMN2
SCHEMBL5309136 0.85 CA12 (0.40) TP53RXFP1NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007039146-A1 4-CARBOXY PYRAZOLE DERIVATIVES AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2007-04-12 WO disclosed
WO-2007039146-A1 4-CARBOXY PYRAZOLE DERIVATIVES AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2007-04-12 WO disclosed