SCHEMBL5309237

SCHEMBL5309237

COc1cnc(Cl)nc1N(CC(C)C)NC(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
STK17B O94768 1/20 0.40
STK17A Q9UEE5 1/20 0.40
AAK1 Q2M2I8 17/20 0.39
TRPA1 O75762 1/20 0.34
ATR Q13535 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3316282 0.88 STK17B (0.41) STK17BSTK17AAAK1TRPA1
SCHEMBL5306326 0.88 STK17B (0.47) STK17BSTK17AAAK1TRPA1ATR
SCHEMBL5792631 0.87 STK17B (0.42) STK17BSTK17AAAK1TRPA1
SCHEMBL5306991 0.86 STK17B (0.41) STK17BSTK17AAAK1TRPA1
SCHEMBL8245020 0.84 CTSL (0.43) AAK1
SCHEMBL5306740 0.82 STK17B (0.39) STK17BSTK17AAAK1TRPA1
SCHEMBL5306935 0.78 AAK1 (0.36) STK17BSTK17AAAK1
SCHEMBL8243205 0.77 STK17B (0.40) STK17BSTK17AAAK1TRPA1ATR
SCHEMBL8140939 0.76 AAK1 (0.47) STK17BSTK17AAAK1TRPA1ATR
SCHEMBL30068217 0.76 ALDH1A1 (0.38) STK17BSTK17AAAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025776-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed
WO-2007025776-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed