SCHEMBL5309369

SCHEMBL5309369

N#Cc1cnc2c(ccc3[nH]nnc32)c1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 2/20 0.44
IMPDH2 P12268 1/20 0.36
IMPDH1 P20839 1/20 0.36
CCR1 P32246 2/20 0.33
CCR5 P51681 2/20 0.33
CCR8 P51685 2/20 0.33
SLC40A1 Q9NP59 1/20 0.33
CYP19A1 P11511 2/20 0.33
HTT P42858 1/20 0.33
LRRK2 Q5S007 1/20 0.32
METAP2 P50579 1/20 0.32
PARP1 P09874 2/20 0.32
CYP11B1 P15538 2/20 0.31
CYP11B2 P19099 2/20 0.31
TRPA1 O75762 1/20 0.31
MAP3K14 Q99558 1/20 0.31
VCP P55072 1/20 0.31
CYP17A1 P05093 1/20 0.31
CHUK O15111 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11910642 0.82 HPGDS (0.59) HPGDSIMPDH2IMPDH1CCR1CCR5
SCHEMBL30492619 0.82 HPGDS (0.59) HPGDSIMPDH2IMPDH1CCR1CCR5
SCHEMBL5310535 0.77 HPGDS (0.46) HPGDSIMPDH2IMPDH1CCR1CCR5
SCHEMBL5314035 0.75 HPGDS (0.43) HPGDSIMPDH2IMPDH1CYP19A1HTT
SCHEMBL1994732 0.74 CCR1 (0.57) HPGDSCCR1CCR5CCR8SLC40A1
SCHEMBL30492680 0.74 CCR1 (0.57) HPGDSCCR1CCR5CCR8SLC40A1
SCHEMBL5251543 0.72 ALDH1A1 (0.43) TRPA1
SCHEMBL5260083 0.71 HPGDS (0.43) HPGDSIMPDH2IMPDH1CYP19A1HTT
SCHEMBL5260088 0.71 HPGDS (0.43) HPGDSIMPDH2IMPDH1HTT
SCHEMBL11910090 0.69 HPGDS (0.47) HPGDSCCR1CCR5CCR8HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242382-B1 TRICYCLIC PROTEIN KINASE INHIBITORS WYETH CORP (US) 2007-02-07 EP claimed