SCHEMBL5310013

SCHEMBL5310013

Cn1nc(-c2ccc(C(=O)CC#N)cc2)cc1C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 2/20 0.43
HDAC4 P56524 2/20 0.43
HDAC1 Q13547 2/20 0.43
HDAC7 Q8WUI4 2/20 0.43
HDAC2 Q92769 2/20 0.43
HDAC10 Q969S8 2/20 0.43
HDAC11 Q96DB2 2/20 0.43
HDAC8 Q9BY41 2/20 0.43
HDAC6 Q9UBN7 2/20 0.43
HDAC9 Q9UKV0 2/20 0.43
HDAC5 Q9UQL6 2/20 0.43
NCOR2 Q9Y618 2/20 0.43
ALDH1A1 P00352 4/20 0.43
PKM P14618 1/20 0.42
SCN9A Q15858 1/20 0.40
RXFP1 Q9HBX9 1/20 0.39
GAA P10253 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5306702 0.80 ALDH1A1 (0.49) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL1593804 0.77 ALDH1A1 (0.62) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL1594334 0.75 ALDH1A1 (0.42) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL1595751 0.73 HPGD (0.53) HDAC4HDAC6ALDH1A1PKMNPC1
SCHEMBL5307103 0.72 ALDH1A1 (0.50) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL21611649 0.72 NPC1 (0.55) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL5303980 0.71 ALDH1A1 (0.44) ALDH1A1PKMGAAL3MBTL1NPC1
SCHEMBL13098615 0.71 KEAP1 (0.47) ALDH1A1PKMGAAL3MBTL1NPC1
SCHEMBL5307435 0.71 TP53 (0.57) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL13098073 0.71 TP53 (0.59) ALDH1A1L3MBTL1NPC1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007034279-A2 C3A ANTAGONISTS AND PHARMACEUTICAL COMPOSITIONS THEREOF PFIZER PRODUCTS INC. (US) 2007-03-29 WO disclosed