SCHEMBL5310014

SCHEMBL5310014

CNC(=O)c1ccc(N2C=CCN(C(=O)c3cc(F)ccc3C(F)(F)F)C2=O)nc1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BRAF P15056 5/20 0.39
KDR P35968 5/20 0.39
PARP1 P09874 1/20 0.38
PTK2 Q05397 1/20 0.36
SCD O00767 3/20 0.36
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
RXRA P19793 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
NTRK1 P04629 1/20 0.35
EGLN1 Q9GZT9 1/20 0.35
KIT P10721 2/20 0.35
FLT3 P36888 2/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
ACSS2 Q9NR19 1/20 0.34
MAPK3 P27361 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5311282 0.91 SCD (0.38) SCDHCRTR1HCRTR2EGLN1
SCHEMBL5307539 0.88 SCD (0.47) BRAFKDRPARP1SCD
SCHEMBL5313445 0.87 KCNQ3 (0.43) BRAFKDRSCD
SCHEMBL5310009 0.83 PARP1 (0.41) BRAFKDRPARP1PTK2SCD
SCHEMBL5307080 0.81 SCD (0.40) BRAFKDRPARP1PTK2SCD
SCHEMBL5309153 0.81 CYP1A2 (0.43) SCD
SCHEMBL5309835 0.79 SCD (0.51) SCDEGLN1
SCHEMBL5306454 0.78 EGLN1 (0.39) EGLN1KDM4EALDH1A1
SCHEMBL5309661 0.78 SCD (0.53) SCDEGLN1
SCHEMBL5311209 0.77 RAB9A (0.38) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007046867-A2 PIPERIDINE DERIVATIVES AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2007-04-26 WO disclosed