SCHEMBL5310036

SCHEMBL5310036

Nc1cccn2cc(-c3ccc(Br)cc3)nc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 13/20 0.60
NPC1 O15118 12/20 0.60
ALDH1A1 P00352 7/20 0.60
MAPT P10636 5/20 0.60
POLB P06746 2/20 0.60
KMT2A Q03164 2/20 0.60
MEN1 O00255 1/20 0.60
APEX1 P27695 1/20 0.60
MAPK1 P28482 1/20 0.60
HTT P42858 1/20 0.60
CTDSP1 Q9GZU7 1/20 0.60
TDP1 Q9NUW8 1/20 0.60
KDM4E B2RXH2 8/20 0.56
TP53 P04637 3/20 0.54
HSD17B10 Q99714 3/20 0.54
GAA P10253 3/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
HPGD P15428 2/20 0.54
NFKB1 P19838 2/20 0.51
NFKB2 Q00653 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9082442 0.85 ALDH1A3 (0.68) RAB9ANPC1ALDH1A1MAPTKMT2A
SCHEMBL19322146 0.81 NPC1 (0.60) RAB9ANPC1ALDH1A1MAPTPOLB
SCHEMBL972723 0.81 NPC1 (0.77) RAB9ANPC1ALDH1A1MAPTPOLB
Bromide SCHEMBL1691886 0.80 NPC1 (0.75) RAB9ANPC1ALDH1A1MAPTPOLB
SCHEMBL5852628 0.79 DHODH (0.63) RAB9ANPC1ALDH1A1MAPTPOLB
Bromide SCHEMBL8866070 0.79 DHODH (0.59) RAB9ANPC1ALDH1A1MAPTPOLB
SCHEMBL14542378 0.78 NPC1 (0.56) RAB9ANPC1ALDH1A1MAPTPOLB
SCHEMBL18038275 0.78 DHODH (0.79) RAB9ANPC1ALDH1A1MAPTPOLB
SCHEMBL1420335 0.76 ALDH1A3 (0.55) RAB9ANPC1ALDH1A1POLBKDM4E
SCHEMBL5313388 0.76 NPC1 (1.00) RAB9ANPC1ALDH1A1MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007039146-A1 4-CARBOXY PYRAZOLE DERIVATIVES AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2007-04-12 WO disclosed
WO-2007039146-A1 4-CARBOXY PYRAZOLE DERIVATIVES AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2007-04-12 WO disclosed