SCHEMBL5313388

SCHEMBL5313388

O=[N+]([O-])c1cccn2cc(-c3ccc(Br)cc3)nc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 13/20 1.00
RAB9A P51151 13/20 1.00
ALDH1A1 P00352 9/20 1.00
MAPT P10636 6/20 1.00
POLB P06746 3/20 1.00
HTT P42858 2/20 1.00
MEN1 O00255 1/20 1.00
APEX1 P27695 1/20 1.00
MAPK1 P28482 1/20 1.00
KMT2A Q03164 1/20 1.00
CTDSP1 Q9GZU7 1/20 1.00
TDP1 Q9NUW8 1/20 1.00
HRH3 Q9Y5N1 1/20 0.56
KDM4E B2RXH2 7/20 0.50
SMN1; SMN2 Q16637 5/20 0.48
TP53 P04637 3/20 0.48
HSD17B10 Q99714 3/20 0.48
GAA P10253 3/20 0.48
HPGD P15428 2/20 0.48
DHODH Q02127 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5738629 0.86 NPC1 (0.76) NPC1RAB9AALDH1A1MAPTPOLB
SCHEMBL1420384 0.79 NPC1 (0.65) NPC1RAB9AALDH1A1MAPTPOLB
SCHEMBL19322146 0.76 NPC1 (0.60) NPC1RAB9AALDH1A1MAPTPOLB
SCHEMBL972723 0.76 NPC1 (0.77) NPC1RAB9AALDH1A1MAPTPOLB
SCHEMBL5310036 0.76 RAB9A (0.60) NPC1RAB9AALDH1A1MAPTPOLB
SCHEMBL1419901 0.75 MAPT (0.60) NPC1RAB9AALDH1A1MAPTPOLB
SCHEMBL18038275 0.75 DHODH (0.79) NPC1RAB9AALDH1A1MAPTPOLB
Bromide SCHEMBL1691886 0.74 NPC1 (0.75) NPC1RAB9AALDH1A1MAPTPOLB
SCHEMBL9096250 0.74 ALDH1A1 (0.58) NPC1RAB9AALDH1A1MAPTPOLB
SCHEMBL5852628 0.73 DHODH (0.63) NPC1RAB9AALDH1A1MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007039146-A1 4-CARBOXY PYRAZOLE DERIVATIVES AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2007-04-12 WO disclosed