SCHEMBL531061

SCHEMBL531061

CCCCCCNC(C)C(=O)c1cnc2ccccc2c1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 13/20 0.49
MGAM O43451 1/20 0.47
HDAC3 O15379 2/20 0.45
HDAC1 Q13547 2/20 0.45
HDAC2 Q92769 1/20 0.45
CCKBR P32239 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5020897 0.79 HDAC3 (0.61) TRPV1MGAMHDAC3HDAC1HDAC2
SCHEMBL12505087 0.79 TRPV1 (0.51) TRPV1MGAMHDAC3HDAC1HDAC2
SCHEMBL11416534 0.77 NAAA (0.55) HDAC3HDAC1HDAC2
SCHEMBL10242977 0.75 HDAC3 (0.61) TRPV1MGAMHDAC3HDAC1HDAC2
SCHEMBL2625196 0.75 MGAM (0.65) TRPV1MGAM
SCHEMBL531058 0.74 NAAA (0.50) TRPV1HDAC3HDAC1HDAC2
SCHEMBL12505086 0.74 TRPV1 (0.43) TRPV1HDAC3HDAC1HDAC2
SCHEMBL13610181 0.73 LMNA (0.55) TRPV1MGAM
SCHEMBL27391699 0.73 LMNA (0.55) TRPV1MGAM
SCHEMBL9360308 0.73 MGAM (0.58) TRPV1MGAMHDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed