SCHEMBL5310850

SCHEMBL5310850

Cc1ccccc1OC(=O)C(O)(c1ccccc1C)C(O)C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
PPARG P37231 1/20 0.38
BCHE P06276 1/20 0.35
KDM4E B2RXH2 2/20 0.35
GAA P10253 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ELANE P08246 2/20 0.35
CYP1A2 P05177 1/20 0.34
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34
NOTUM Q6P988 1/20 0.34
HTT P42858 1/20 0.34
CASP1 P29466 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12817104 0.81 CPT2 (0.35) ATMTDP1L3MBTL1KDM4EGAA
SCHEMBL697581 0.81 CPT2 (0.35) ATMTDP1L3MBTL1KDM4EGAA
Water SCHEMBL28155256 0.79 CPT2 (0.34) ATMTDP1L3MBTL1KDM4EGAA
SCHEMBL689263 0.79 GAA (0.35) ATMTDP1PPARGKDM4EGAA
SCHEMBL27524735 0.74 SLC1A3 (0.36) TDP1L3MBTL1KDM4EGAAALDH1A1
SCHEMBL4668126 0.73 KDM4E (0.38) ATMTDP1L3MBTL1PPARGKDM4E
SCHEMBL1162260 0.73 KDM4E (0.38) ATMTDP1L3MBTL1PPARGKDM4E
SCHEMBL555425 0.73 KDM4E (0.38) ATMTDP1L3MBTL1PPARGKDM4E
SCHEMBL15538386 0.72 GABRA1 (0.36) ATMTDP1L3MBTL1KDM4EGAA
SCHEMBL15539622 0.72 GABRA1 (0.36) ATMTDP1L3MBTL1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102351918-B Glucopyranosyl-substituted benzonitrile derivatives and pharmaceutical compositions containing the same BOEHRINGER INGELHEIM INT 2015-03-04 CN disclosed
CN-103601709-A Glucopyranosyl-substituted benzonitrile derivatives, pharmaceutical compositions containing such compounds, their use and process for their manufacture BOEHRINGER INGELHEIM INT 2014-02-26 CN disclosed
CN-101939316-B Spirocyclic heterocyclic compounds, medicaments containing said compounds, their use and processes for their preparation BOEHRINGER INGELHEIM INT 2013-10-02 CN disclosed
CN-102351918-A Glucopyranosyl-substituted benzonitrile derivatives, pharmaceutical compositions containing said compounds, their use and process for their preparation BOEHRINGER INGELHEIM INT 2012-02-15 CN disclosed
CN-102203064-A Novel benzamides, their preparation and their use as medicaments BOEHRINGER INGELHEIM INT 2011-09-28 CN disclosed
CN-101437807-A Glucopyranosyl-substituted benzonitrile derivatives, pharmaceutical compositions containing said compounds, their use and process for their preparation BOEHRINGER INGELHEIM INT (DE) 2009-05-20 CN disclosed
CN-101384576-A Glucopyranosyl-substituted benzonitrile derivatives, pharmaceutical compositions containing such compounds, their use and process for their manufacture BOEHRINGER INGELHEIM INT (DE) 2009-03-11 CN disclosed
WO-2007052134-A1 (2S)-2-AMINOMETHYL-5-ETHYL HEPTANOIC ACID ITS PHARMACEUTICAL USE PFIZER LIMITED (GB) 2007-05-10 WO disclosed
CN-1880312-A Alkoxy substituted benzimidazole compounds, pharmaceutical preparations containing the same AAIPHARMA INC (US) 2006-12-20 CN disclosed
WO-2006092692-A1 USE OF COMBINATIONS OF PDE7 INHIBITORS AND ALPHA-2-DELTY LIGANDS FOR THE TREATMENT OF NEUROPATHIC PAIN PFIZER LIMITED (GB) 2006-09-08 WO disclosed
CN-1183127-C Alkoxy-substituted benzimidazole compounds, pharmaceutical formulations containing them and methods of using them 2005-01-05 CN disclosed
CN-1509270-A Indolinones substituted in the 6-position, process for their preparation and their use as kinase inhibitors ���ָ��Ӣ��ķ�������Ϲ�˾ 2004-06-30 CN disclosed
CN-1384831-A Alkoxy-substituted benzimidazole compounds, pharmaceutical formulations containing them and methods of using them EIPHAVMA INC (US) 2002-12-11 CN disclosed
CN-1319090-A Novel substuted indolimones, their preparation process and use as medicine BOEHRINGER INGELHEIM PHARMA (DE) 2001-10-24 CN disclosed
CN-1187186-A Substituted phenyl amindines, medicaments containing these compounds and process for producing them THOMAE GMBH DR K (DE) 1998-07-08 CN disclosed
CN-1087904-A Carboxylic acid derivative, the pharmaceutical composition that contains these compounds with and preparation method thereof KRAL THOMAE GMBH (DE) 1994-06-15 CN disclosed