SCHEMBL5311319

SCHEMBL5311319

C[C@@](NC(=O)c1ccc(-c2ccc(C(F)(F)F)cc2)cc1)(C(=O)O)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.51
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
HDAC2 Q92769 1/20 0.47
CTDSP1 Q9GZU7 1/20 0.46
TRPV1 Q8NER1 1/20 0.46
DRD2 P14416 1/20 0.45
DRD4 P21917 1/20 0.45
CYP3A4 P08684 1/20 0.44
PTPN5 P54829 1/20 0.44
CHRM4 P08173 1/20 0.44
BACE1 P56817 1/20 0.44
PTGS1 P23219 1/20 0.43
CRHBP P24387 1/20 0.43
CRHR2 Q13324 1/20 0.43
TMEM97 Q5BJF2 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28250048 0.93 RAB9A (0.51) NPC1RAB9ATRPV1PTGS1CRHBP
SCHEMBL28250047 0.91 NPC1 (0.57) NPC1RAB9AHDAC2TRPV1PTGS1
SCHEMBL28536704 0.90 CTDSP1 (0.53) NPC1RAB9ACTDSP1MAPT
SCHEMBL28250190 0.81 POLB (0.54) NPC1RAB9AHDAC2CYP3A4
SCHEMBL28250050 0.80 KCNK3 (0.55) NPC1RAB9AMAPT
SCHEMBL28908852 0.78 POLB (0.53) NPC1RAB9ATMEM97SIGMAR1MAPT
SCHEMBL28250847 0.77 NPC1 (0.53) NPC1RAB9AMAPT
SCHEMBL28456845 0.77 TRPV1 (0.54) NPC1RAB9ATRPV1PTGS1
SCHEMBL14714456 0.77 NPC1 (0.56) NPC1RAB9AHDAC2CTDSP1DRD2
SCHEMBL6416083 0.76 NPC1 (0.60) NPC1RAB9ACTDSP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007044574-A2 PHARMACEUTICAL COMPOSITIONS, METHODS OF PREPARATION THEREOF, AND METHODS OF TREATMENT TRANSTECH PHARMA, INC. (US) 2007-04-19 WO disclosed
US-20070082952-A1 Pharmaceutical compositions, methods of preparation thereof, and methods of treatment TRANSTECH PHARMA, INC. 2007-04-12 US disclosed