SCHEMBL5311552

SCHEMBL5311552

COc1ccccc1-c1c(C)nn(C(C)C)c(=O)c1CCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.48
PDE1A P54750 2/20 0.43
PDE1B Q01064 2/20 0.43
PDE1C Q14123 2/20 0.43
TP53 P04637 2/20 0.41
TSHR P16473 2/20 0.39
MAPT P10636 5/20 0.39
ALDH1A1 P00352 4/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
HPGD P15428 3/20 0.39
PLAT P00750 1/20 0.38
GNRHR P30968 1/20 0.37
HSD17B10 Q99714 1/20 0.37
USP2 O75604 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5311895 0.89 GNRHR (0.42) KDM4EPDE1APDE1BPDE1CTSHR
SCHEMBL5311130 0.86 KDM4E (0.42) KDM4EPDE1APDE1BPDE1CTP53
SCHEMBL5311949 0.84 CASR (0.47) KDM4EUSP2POLBPDE4APDE4B
SCHEMBL5311530 0.82 GNRHR (0.49) GNRHR
SCHEMBL5310470 0.82 KDM4E (0.41) KDM4ETP53MAPTGNRHRCYP3A4
SCHEMBL5315640 0.80 BRD4 (0.40) KDM4ETSHRMAPTALDH1A1CYP1A2
SCHEMBL5313086 0.77 GNRHR (0.40) KDM4EMAPTGNRHRTHRB
SCHEMBL5311941 0.76 GNRHR (0.40) MAPTGNRHR
SCHEMBL5313183 0.76 PDE1A (0.43) KDM4EPDE1APDE1BPDE1CTP53
SCHEMBL5313180 0.76 PDE1A (0.43) KDM4EPDE1APDE1BPDE1CTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007044796-A2 PYRIDAZINONE COMPOUNDS AS CALCILYTICS NPS PHARMACEUTICALS, INC. (US) 2007-04-19 WO disclosed
WO-2007044796-A2 PYRIDAZINONE COMPOUNDS AS CALCILYTICS NPS PHARMACEUTICALS, INC. (US) 2007-04-19 WO disclosed