SCHEMBL5312450

SCHEMBL5312450

CC(=O)OC(C)(Cc1cc(Br)c(OCc2cccc(NS(C)(=O)=O)c2Cl)c(Br)c1)C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRA P10827 8/20 0.38
THRB P10828 8/20 0.38
SLC16A3 O15427 1/20 0.34
SLC16A1 P53985 1/20 0.34
MCTS1 Q9ULC4 1/20 0.34
NR3C1 P04150 4/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2C19 P33261 2/20 0.33
NR3C2 P08235 2/20 0.33
CYP2C9 P11712 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ESR1 P03372 1/20 0.33
PGR P06401 1/20 0.33
AR P10275 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
RCE1 Q9Y256 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5116725 0.80 THRA (0.60) THRATHRBNR3C1NR3C2ESR1
SCHEMBL5310031 0.79 THRA (0.41) THRATHRBNR3C1CYP1A2CYP3A4
SCHEMBL5311039 0.78 THRA (0.40) THRATHRBNR3C1CYP1A2CYP3A4
SCHEMBL4356784 0.78 THRA (0.40) THRATHRBNR3C1CYP1A2CYP3A4
SCHEMBL5308746 0.77 THRA (0.36) THRATHRBNR3C1CYP1A2CYP3A4
SCHEMBL14540614 0.76 THRA (0.38) THRATHRBNR3C1CYP1A2CYP3A4
SCHEMBL5310191 0.76 THRA (0.38) THRATHRBNR3C1CYP1A2CYP3A4
SCHEMBL5309606 0.76 THRA (0.38) THRATHRBNR3C1CYP1A2CYP3A4
SCHEMBL5111310 0.72 THRA (0.59) THRATHRBNR3C1NR3C2ESR1
SCHEMBL5112565 0.71 THRA (0.63) THRATHRBNR3C1NR3C2ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007039125-A2 AN OPTICALLY ACTIVE THYROID RECEPTOR AGONIST AND OPTICALLY ACTIVE KEY INTERMEDIATES IN ITS PRODUCTION KARO BIO AB (SE) 2007-04-12 WO disclosed