SCHEMBL5310031

SCHEMBL5310031

CS(=O)(=O)Nc1cccc(COc2c(Br)cc(CC(O)C(=O)O)cc2Br)c1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRA P10827 7/20 0.41
THRB P10828 7/20 0.41
NR3C1 P04150 3/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C19 P33261 2/20 0.36
ESR1 P03372 1/20 0.35
PGR P06401 1/20 0.35
NR3C2 P08235 1/20 0.35
AR P10275 1/20 0.35
CYP2C9 P11712 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PPARG P37231 1/20 0.35
FABP4 P15090 2/20 0.35
FABP5 Q01469 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
RCE1 Q9Y256 1/20 0.35
PDCD1 Q15116 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5310191 0.91 THRA (0.38) THRATHRBNR3C1CYP1A2CYP3A4
SCHEMBL4356784 0.89 THRA (0.40) THRATHRBNR3C1CYP1A2CYP3A4
SCHEMBL5311039 0.89 THRA (0.40) THRATHRBNR3C1CYP1A2CYP3A4
SCHEMBL5309606 0.85 THRA (0.38) THRATHRBNR3C1CYP1A2CYP3A4
SCHEMBL14540614 0.85 THRA (0.38) THRATHRBNR3C1CYP1A2CYP3A4
SCHEMBL5116725 0.84 THRA (0.60) THRATHRBNR3C1ESR1PGR
SCHEMBL5308746 0.82 THRA (0.36) THRATHRBNR3C1CYP1A2CYP3A4
SCHEMBL5312450 0.79 THRA (0.38) THRATHRBNR3C1CYP1A2CYP3A4
SCHEMBL14541012 0.77 THRA (0.41) THRATHRBNR3C1ESR1PGR
SCHEMBL4345797 0.77 THRB (0.34) THRATHRBCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007039125-A2 AN OPTICALLY ACTIVE THYROID RECEPTOR AGONIST AND OPTICALLY ACTIVE KEY INTERMEDIATES IN ITS PRODUCTION KARO BIO AB (SE) 2007-04-12 WO disclosed