SCHEMBL5312970

SCHEMBL5312970

O=C1NC(=O)c2c(CCCCl)cccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.41
ALDH1A1 P00352 4/20 0.40
KDM4E B2RXH2 4/20 0.40
GAA P10253 2/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
PARP1 P09874 4/20 0.39
CASP3 P42574 6/20 0.37
MAPT P10636 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
RAB9A P51151 1/20 0.37
SENP8 Q96LD8 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
RXFP1 Q9HBX9 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CASP7 P55210 2/20 0.36
CASP2 P42575 1/20 0.36
CASP6 P55212 1/20 0.36
CASP8 Q14790 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8969034 0.95 PARP1 (0.42) GSK3BALDH1A1KDM4EGAAHPGD
SCHEMBL10354541 0.90 GSK3B (0.43) GSK3BALDH1A1KDM4EGAAHPGD
SCHEMBL10914947 0.88 GSK3B (0.45) GSK3BALDH1A1KDM4EGAAHPGD
SCHEMBL10712855 0.88 GSK3B (0.45) GSK3BALDH1A1KDM4EGAAHPGD
SCHEMBL11206986 0.88 GSK3B (0.45) GSK3BALDH1A1KDM4EGAAHPGD
SCHEMBL11015946 0.88 GSK3B (0.45) GSK3BALDH1A1KDM4EGAAHPGD
SCHEMBL5970012 0.86 GSK3B (0.50) GSK3BALDH1A1KDM4EGAAHPGD
SCHEMBL4343595 0.83 GSK3B (0.41) GSK3BALDH1A1KDM4EGAAHPGD
SCHEMBL335247 0.83 GSK3B (0.41) GSK3BALDH1A1KDM4EGAAHPGD
SCHEMBL166776 0.83 ELANE (0.43) GSK3BALDH1A1KDM4EGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007058630-A1 NOVEL BIS(AMINO)-ORTHO-DICARBABORANE CLUSTER COMPOUNDS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2007-05-24 WO disclosed
US-5585392-A TREATING OR PREVENTING STROKES BAYER AKTIENGESELLSCHAFT (DE) 1996-12-17 US disclosed
US-5506246-A Method for treating depression using substituted aminomethyltetralins and their heterocyclic analogues BAYER AKTIENGESELLSCHAFT (DE) 1996-04-09 US disclosed
US-5463105-A Therapy for cardiovascular, nervous system disorders BAYER AKTIENGESELLSCHAFT (DE) 1995-10-31 US disclosed
EP-0231159-B1 Indoloquinoxalines with substituents in 6-position containing cyclic groups LUNDBLAD LEIF (SE) 1994-08-10 EP disclosed
EP-0352613-B1 Substituted amino methyl tetralines, and their heterocyclic analogous compounds BAYER AG (DE) 1994-04-20 EP disclosed
US-5298513-A Serotonin antagonist BAYER AKTIENGESELLSCHAFT (DE) 1994-03-29 US disclosed
EP-0332968-B1 1,3,4,5-Tetrahydrobenz[c,d]indoles BAYER AG (DE) 1993-06-02 EP disclosed
US-5153225-A For treating disorders of the central nervous system, cardiovascular system and intestinal tract BAYER AKTIENGESELLSCHAFT (DE) 1992-10-06 US disclosed
US-5137901-A For binding 5-HT 1 receptors; treating central nervous system disorders BAYER AKTIENGESELLSCHAFT (DE) 1992-08-11 US disclosed
US-4990510-A Viricides, anticancer agents LEIF LUNDBLAD (BE) 1991-02-05 US disclosed
EP-0390515-A1 Novel adenine derivatives and their use as agents for increasing crop yields MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 1990-10-03 EP disclosed
US-4916124-A Indoloquinoxalines with substituents in 6-position containing cyclic groups as antiviral agents Lundblad, Lief (SE) 1990-04-10 US disclosed
EP-0352613-A2 Substituted amino methyl tetralines, and their heterocyclic analogous compounds BAYER AG (DE) 1990-01-31 EP disclosed
US-4880802-A CENTRAL NERVOUS SYSTEM BAYER AKTIENGESELLSCHAFT (DE) 1989-11-14 US disclosed
EP-0332968-A1 1,3,4,5-Tetrahydrobenz[c,d]indoles BAYER AG (DE) 1989-09-20 EP disclosed
EP-0270947-A2 Substituted basic 2-aminotetralines BAYER AG (DE) 1988-06-15 EP disclosed
EP-0238459-A1 Substituted indoloquinoxalines Lundblad, Leif (SE) 1987-09-23 EP disclosed
EP-0231159-A1 Indoloquinoxalines with substituents in 6-position containing cyclic groups Lundblad, Leif (SE) 1987-08-05 EP disclosed
WO-1987004436-A1 SUBSTITUTED INDOLOQUINOXALINES LUNDBLAD, LEIF (SE) 1987-07-30 WO disclosed