SCHEMBL5312975

SCHEMBL5312975

Cc1csc(-n2c(C)ccc2-c2ccc(S(N)(=O)=O)cc2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.46
CA1 P00915 8/20 0.44
CA2 P00918 8/20 0.44
CA9 Q16790 8/20 0.44
CA12 O43570 7/20 0.44
PTGS1 P23219 4/20 0.41
CA3 P07451 2/20 0.40
CA6 P23280 2/20 0.40
CA5A P35218 2/20 0.40
CA7 P43166 2/20 0.40
CA5B Q9Y2D0 2/20 0.40
CHRNA7 P36544 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
PTGES O14684 1/20 0.39
HDAC3 O15379 1/20 0.39
PDPK1 O15530 1/20 0.39
PDE5A O76074 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7216716 0.88 PTGS2 (0.60) PTGS2PTGS1KDM4EALDH1A1MAPT
SCHEMBL2465765 0.87 CA12 (0.42) PTGS2CA1CA2CA9CA12
SCHEMBL348164 0.80 CA2 (0.44) PTGS2CA1CA2CA9CA12
SCHEMBL5315712 0.78 PTGS2 (0.52) PTGS2CA1CA2CA9CA12
SCHEMBL8504980 0.77 CA2 (0.35) PTGS2CA1CA2CA9CA12
SCHEMBL7210840 0.76 PTGS2 (0.76) PTGS2CA1CA2CA9CA12
SCHEMBL7216218 0.73 PTGS2 (0.76) PTGS2CA1CA2CA9CA12
SCHEMBL3690377 0.73 PTGS2 (0.41) PTGS2CA1CA2CA9CA12
SCHEMBL27767202 0.72 PTGS2 (0.57) PTGS2CA1CA2CA9CA12
SCHEMBL3025180 0.71 PTGS2 (0.68) PTGS2CA1CA2CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799823-B1 1,2-Diphenylpyrrole derivatives, their preparation and their therapeutic uses DAIICHI SANKYO CO LTD (JP) 2007-10-31 EP disclosed
US-RE39420-E1 1,2-Diphenylpyrrole derivatives, their preparation and their therapeutic uses SANKYO COMPANY, LIMITED (JP) 2006-12-05 US disclosed
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP disclosed
US-5908858-A OSTEOPOROSIS; LEUKOTRIENE INHIBITOR SANKYO COMPANY, LIMITED (JP) 1999-06-01 US disclosed
EP-0799823-A1 1,2-Diphenylpyrrole derivatives, their preparation and their therapeutic uses SANKYO COMPANY LIMITED (JP) 1997-10-08 EP disclosed