SCHEMBL5313574

SCHEMBL5313574

O=Cc1conc1-c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.45
GSR P00390 1/20 0.45
KMT2A Q03164 4/20 0.39
MEN1 O00255 3/20 0.39
LMNA P02545 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
THRB P10828 1/20 0.39
BLM P54132 1/20 0.39
HSP90AA1 P07900 1/20 0.39
TP53 P04637 1/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ALDH1A1 P00352 2/20 0.38
NPC1 O15118 2/20 0.38
POLB P06746 2/20 0.38
KDM4E B2RXH2 1/20 0.38
PTPN1 P18031 3/20 0.37
PTPN2 P17706 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4973045 0.73 PTGS2 (0.41) PTGS2GSRKMT2AMEN1LMNA
SCHEMBL27442348 0.73 PTGS2 (0.41) PTGS2GSRKMT2AMEN1LMNA
SCHEMBL1797330 0.71 PTGS2 (0.67) PTGS2KMT2AMEN1LMNATDP1
SCHEMBL4975519 0.70 PTGS2 (0.39) PTGS2GSRKMT2AMEN1LMNA
SCHEMBL27813684 0.69 PTGS2 (0.47) PTGS2KMT2AMEN1LMNATDP1
SCHEMBL1092219 0.69 CYP19A1 (0.53) PTGS2KMT2AMEN1LMNATDP1
SCHEMBL3658890 0.69 HSP90AA1 (0.54) PTGS2KMT2AMEN1LMNATDP1
SCHEMBL5425872 0.69 PTGS2 (0.47) PTGS2KMT2AMEN1LMNATDP1
SCHEMBL27217198 0.69 PTGS2 (0.44) PTGS2KMT2AMEN1LMNATDP1
SCHEMBL27514872 0.69 PTGS2 (0.44) PTGS2KMT2AMEN1LMNATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765795-A2 ALKYNYL DERIVATIVES AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS Addex Pharmaceuticals SA (CH) 2007-03-28 EP disclosed
WO-2005123703-A2 ALKYNYL DERIVATIVES AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS ADDEX PHARMACEUTICALS SA (CH) 2005-12-29 WO disclosed