SCHEMBL4973045

SCHEMBL4973045

O=CCc1conc1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.41
GABRA5 P31644 2/20 0.40
GSR P00390 1/20 0.38
HSP90AA1 P07900 1/20 0.36
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
NOTUM Q6P988 1/20 0.34
CA12 O43570 2/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA9 Q16790 2/20 0.33
PTGS1 P23219 2/20 0.33
NR4A2 P43354 1/20 0.33
FFAR4 Q5NUL3 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23366325 0.80 PTGS2 (0.47) PTGS2GABRA5HSP90AA1MEN1LMNA
SCHEMBL11848234 0.80 PTGS2 (0.39) PTGS2GABRA5GSRHSP90AA1MEN1
SCHEMBL28139688 0.77 NOTUM (0.44) PTGS2GABRA5HSP90AA1MEN1LMNA
SCHEMBL8306253 0.77 GABRA5 (0.42) PTGS2GABRA5HSP90AA1MEN1LMNA
SCHEMBL2929388 0.77 NOTUM (0.49) PTGS2GABRA5HSP90AA1MEN1LMNA
SCHEMBL3213310 0.77 PTGS2 (0.41) PTGS2GABRA5GSRHSP90AA1MEN1
SCHEMBL27819710 0.76 KDM4E (0.49) PTGS2GABRA5HSP90AA1LMNAHTT
SCHEMBL5775916 0.74 NOTUM (0.46) PTGS2GABRA5HSP90AA1MEN1LMNA
SCHEMBL5772931 0.74 PTGS2 (0.42) PTGS2GABRA5GSRHSP90AA1MEN1
SCHEMBL5313574 0.73 PTGS2 (0.45) PTGS2GSRHSP90AA1MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968973-A2 ARYL-ISOXAZOL-4-YL-IMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2008-09-17 EP disclosed
WO-2007074078-A2 ARYL-ISOXAZOL-4-YL-IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-07-05 WO disclosed