SCHEMBL5314566

SCHEMBL5314566

Cn1ncc(-c2ccnc(NC3CNC3)n2)c1N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 14/20 0.46
CDK2 P24941 7/20 0.46
GSK3B P49841 7/20 0.46
CDK1 P06493 7/20 0.45
CCNB1 P14635 6/20 0.45
CCNA2 P20248 6/20 0.45
CCND1 P24385 5/20 0.45
CCNA1 P78396 5/20 0.45
HRH3 Q9Y5N1 1/20 0.42
RET P07949 1/20 0.42
CCNE1 P24864 2/20 0.42
CCND3 P30281 2/20 0.42
CDK6 Q00534 2/20 0.42
MAPK8 P45983 2/20 0.41
KCNH2 Q12809 1/20 0.41
CCNB2 O95067 1/20 0.41
CCNB3 Q8WWL7 1/20 0.41
MAPK9 P45984 1/20 0.41
MAPK10 P53779 1/20 0.41
MKNK1 Q9BUB5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8227901 0.88 CDK4 (0.57) CDK4CDK2GSK3BCDK1CCNB1
SCHEMBL8235871 0.86 CDK4 (0.58) CDK4CDK2GSK3BCDK1CCNB1
SCHEMBL8233031 0.85 PIK3C3 (0.54) CDK4CDK2GSK3BCDK1CCNB1
SCHEMBL8234846 0.83 CDK4 (0.44) CDK4CDK2GSK3BCDK1CCNB1
SCHEMBL8236676 0.83 CDK2 (0.41) CDK4CDK2GSK3BCDK1CCNB1
SCHEMBL8235108 0.82 CDK4 (0.51) CDK4CDK2GSK3BCDK1CCNB1
SCHEMBL8228339 0.82 MKNK1 (0.50) CDK4CDK2GSK3BRETMAPK8
SCHEMBL8229248 0.81 CDK4 (0.50) CDK4CDK2GSK3BCDK1CCNB1
SCHEMBL8233013 0.80 CDK4 (0.44) CDK4CDK2GSK3BCDK1CCNB1
SCHEMBL8229238 0.80 MAPK8 (0.52) CDK4CDK2GSK3BCDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007129195-A2 4-PYRIMIDINE-5-AMINO-PYRAZOLE COMPOUNDS PFIZER PRODUCTS INC. (US) 2007-11-15 WO disclosed
WO-2007129195-A2 4-PYRIMIDINE-5-AMINO-PYRAZOLE COMPOUNDS PFIZER PRODUCTS INC. (US) 2007-11-15 WO disclosed