SCHEMBL8227901

SCHEMBL8227901

Cn1ncc(-c2ccnc(NC3CCNCC3)n2)c1N

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 11/20 0.57
CDK2 P24941 6/20 0.57
CDK1 P06493 5/20 0.57
CCNB1 P14635 5/20 0.57
CCNA2 P20248 5/20 0.57
CCND1 P24385 5/20 0.57
CCNA1 P78396 5/20 0.57
IKBKB O14920 4/20 0.53
MAPK8 P45983 3/20 0.51
IRAK4 Q9NWZ3 1/20 0.51
GSK3B P49841 6/20 0.50
MKNK1 Q9BUB5 1/20 0.48
FLT3 P36888 1/20 0.45
RET P07949 1/20 0.45
CCNE1 P24864 1/20 0.45
CCND3 P30281 1/20 0.45
CDK6 Q00534 1/20 0.45
KCNH2 Q12809 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5314566 0.88 CDK4 (0.46) CDK4CDK2CDK1CCNB1CCNA2
SCHEMBL8235871 0.88 CDK4 (0.58) CDK4CDK2CDK1CCNB1CCNA2
SCHEMBL8233031 0.87 PIK3C3 (0.54) CDK4CDK2CDK1CCNB1CCNA2
SCHEMBL8229248 0.86 CDK4 (0.50) CDK4CDK2CDK1CCNB1CCNA2
SCHEMBL8235108 0.84 CDK4 (0.51) CDK4CDK2CDK1CCNB1CCNA2
SCHEMBL8228339 0.82 MKNK1 (0.50) CDK4CDK2MAPK8GSK3BMKNK1
SCHEMBL8227898 0.82 IKBKB (0.60) CDK4CDK2CDK1CCNB1CCNA2
SCHEMBL5310500 0.82 CDK4 (0.48) CDK4CDK2CDK1CCNB1CCNA2
SCHEMBL5310502 0.82 CDK4 (0.48) CDK4CDK2CDK1CCNB1CCNA2
SCHEMBL8234846 0.81 CDK4 (0.44) CDK4CDK2CDK1CCNB1CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007129195-A2 4-PYRIMIDINE-5-AMINO-PYRAZOLE COMPOUNDS PFIZER PRODUCTS INC. (US) 2007-11-15 WO disclosed