SCHEMBL5314747

SCHEMBL5314747

CONC(=O)c1cccc(NCc2ccc3nc(Nc4cc(CN(C)C)ccn4)sc3n2)c1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LCK P06239 8/20 0.49
KDR P35968 2/20 0.40
GPR52 Q9Y2T5 3/20 0.38
ROCK1 Q13464 1/20 0.36
ALDH1A1 P00352 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
CDK3 Q00526 1/20 0.34
NOS1 P29475 2/20 0.34
NOS2 P35228 1/20 0.34
ROCK2 O75116 1/20 0.34
GRK2 P25098 1/20 0.34
AURKA O14965 1/20 0.33
RPS6KB1 P23443 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5314803 0.91 LCK (0.40) LCKKDRGPR52ROCK1ALDH1A1
SCHEMBL5314681 0.91 LCK (0.41) LCKKDRGPR52ROCK1ROCK2
SCHEMBL5316017 0.84 KDR (0.51) LCKKDR
SCHEMBL5314751 0.83 LCK (0.50) LCKKDR
SCHEMBL5313953 0.83 KDR (0.51) LCKKDRGPR52ROCK2GRK2
SCHEMBL5314211 0.82 HDAC1 (0.41) LCKKDRALDH1A1ROCK2GRK2
SCHEMBL5315254 0.79 MAPT (0.42) LCKKDRALDH1A1
SCHEMBL5312793 0.78 LCK (0.38) LCKALDH1A1CCNE1CDK2CDK3
SCHEMBL5315698 0.78 LCK (0.38) LCKALDH1A1ROCK2
SCHEMBL5314682 0.75 LCK (0.43) LCKKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007058482-A1 NOVEL INHIBITORS OF PROTEIN KINASE LG LIFE SCIENCES, LTD. (KR) 2007-05-24 WO claimed
WO-2007058482-A1 NOVEL INHIBITORS OF PROTEIN KINASE LG LIFE SCIENCES, LTD. (KR) 2007-05-24 WO disclosed