SCHEMBL5314211

SCHEMBL5314211

CN(C)C(=O)c1cccc(NCc2ccc3nc(Nc4cc(CO)ccn4)sc3n2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
LCK P06239 4/20 0.40
KDR P35968 1/20 0.39
LIPG Q9Y5X9 1/20 0.37
EPHB4 P54760 2/20 0.35
ALDH1A1 P00352 3/20 0.35
CYP3A4 P08684 3/20 0.35
CYP1A2 P05177 2/20 0.35
MAPK1 P28482 2/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TYK2 P29597 1/20 0.35
FYN P06241 4/20 0.35
USP2 O75604 1/20 0.34
CYP2D6 P10635 1/20 0.34
ROCK2 O75116 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5313953 0.89 KDR (0.51) LCKKDRROCK2GRK2
SCHEMBL14530688 0.88 LCK (0.42) LCKLIPGEPHB4ALDH1A1TYK2
SCHEMBL5315254 0.87 MAPT (0.42) LCKKDRALDH1A1CYP1A2HPGD
SCHEMBL5314803 0.82 LCK (0.40) HDAC1HDAC8HDAC6LCKKDR
SCHEMBL5314747 0.82 LCK (0.49) LCKKDRALDH1A1ROCK2GRK2
SCHEMBL5314220 0.82 LCK (0.41) LCKKDRLIPGEPHB4TYK2
SCHEMBL5314681 0.80 LCK (0.41) LCKKDRROCK2GRK2
SCHEMBL5312781 0.78 LCK (0.39) LCKALDH1A1HPGDSMN1; SMN2TYK2
SCHEMBL5315698 0.76 LCK (0.38) LCKALDH1A1HPGDTYK2ROCK2
SCHEMBL5316017 0.74 KDR (0.51) LCKKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007058482-A1 NOVEL INHIBITORS OF PROTEIN KINASE LG LIFE SCIENCES, LTD. (KR) 2007-05-24 WO claimed
WO-2007058482-A1 NOVEL INHIBITORS OF PROTEIN KINASE LG LIFE SCIENCES, LTD. (KR) 2007-05-24 WO disclosed