SCHEMBL5315411

SCHEMBL5315411

[CH2]C(=O)N(C)c1cccc(F)c1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.46
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44
GPBAR1 Q8TDU6 1/20 0.43
PIK3CA P42336 1/20 0.42
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
HTT P42858 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2089025 0.85 CES2 (0.44) PARP1CES2CES1GPBAR1PIK3CA
SCHEMBL2089023 0.85 CES2 (0.44) PARP1CES2CES1GPBAR1PIK3CA
SCHEMBL29460301 0.85 CES2 (0.44) PARP1CES2CES1GPBAR1PIK3CA
SCHEMBL7858429 0.85 CES2 (0.44) PARP1CES2CES1GPBAR1PIK3CA
SCHEMBL10940408 0.83 CES2 (0.42) PARP1CES2CES1GPBAR1PIK3CA
SCHEMBL9956070 0.83 GPBAR1 (0.45) PARP1CES2CES1GPBAR1PIK3CA
SCHEMBL11756402 0.82 BTK (0.46) PARP1CES2CES1GPBAR1PIK3CA
SCHEMBL28250211 0.82 GPBAR1 (0.40) PARP1CES2CES1GPBAR1PIK3CA
Hydrochloric Acid SCHEMBL27945132 0.81 PARP1 (0.47) PARP1CES2CES1GPBAR1PIK3CA
SCHEMBL19027676 0.80 HTT (0.42) CES2CES1GPBAR1PIK3CAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007069986-A1 NEW OXABISPIDINE COMPOUNDS FOR THE TREATMENT OF CARDIAC ARRHYTHMIAS ASTRAZENECA AB (SE) 2007-06-21 WO claimed
WO-2007069986-A1 NEW OXABISPIDINE COMPOUNDS FOR THE TREATMENT OF CARDIAC ARRHYTHMIAS ASTRAZENECA AB (SE) 2007-06-21 WO disclosed