SCHEMBL11756402

SCHEMBL11756402

C=CC(=O)N(C)c1cccc(F)c1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BTK Q06187 5/20 0.46
BRD4 O60885 2/20 0.44
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
PSMB5 P28074 1/20 0.42
PARP1 P09874 1/20 0.41
GPBAR1 Q8TDU6 1/20 0.40
PLCG1 P19174 1/20 0.40
PIK3CA P42336 1/20 0.39
JAK3 P52333 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5315411 0.82 PARP1 (0.46) CES2CES1PARP1GPBAR1PIK3CA
SCHEMBL15088204 0.81 ALDH1A1 (0.53) BTKPLCG1JAK3
SCHEMBL19890630 0.81 HSD17B1 (0.51) BTKJAK3
SCHEMBL23531983 0.81 BTK (0.41) BTKPLCG1JAK3
SCHEMBL29989323 0.80 BTK (0.46) BTKPLCG1JAK3
SCHEMBL7779064 0.80 HTR3E (0.54) BTKGPBAR1
SCHEMBL15974825 0.80 BTK (0.46) BTKPLCG1JAK3
SCHEMBL7535315 0.80 EGFR (0.50) BTKCES2
SCHEMBL10194673 0.79 BCL2A1 (0.49) BRD4
SCHEMBL2089023 0.79 CES2 (0.44) CES2CES1PARP1GPBAR1PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4048018-A Method of carrying out enzyme catalyzed reactions COUGHLIN ROBERT W 1977-09-13 US disclosed
US-4016293-A ADSORBED ON A SUPPORT, CHEESE WHEY COUGHLIN ROBERT W 1977-04-05 US disclosed