SCHEMBL5317431

SCHEMBL5317431

COc1ccc2ncc(Cl)c(CC(O)N3C4CCC3CC(NC/C=C/c3ccccc3)C4)c2c1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.41
MCHR1 Q99705 4/20 0.35
SLC2A1 P11166 1/20 0.35
ALDH1A1 P00352 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
PKM P14618 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5430646 0.83 KCNH2 (0.38) KCNH2MCHR1SLC2A1ALDH1A1L3MBTL1
SCHEMBL5430642 0.83 KCNH2 (0.38) KCNH2MCHR1SLC2A1ALDH1A1L3MBTL1
SCHEMBL3697142 0.76 SLC2A1 (0.47) KCNH2SLC2A1ALDH1A1
SCHEMBL3697147 0.76 SLC2A1 (0.47) KCNH2SLC2A1ALDH1A1
SCHEMBL5317247 0.74 MTNR1A (0.36) KCNH2MCHR1SLC2A1ALDH1A1L3MBTL1
SCHEMBL5317252 0.74 MTNR1A (0.36) KCNH2MCHR1SLC2A1ALDH1A1L3MBTL1
SCHEMBL5728191 0.69 KCNH2 (0.61) KCNH2MCHR1SLC2A1HTR2AHTR2C
SCHEMBL5441471 0.68 KCNH2 (0.40) KCNH2MCHR1SLC2A1ALDH1A1L3MBTL1
SCHEMBL5441479 0.68 KCNH2 (0.40) KCNH2MCHR1SLC2A1ALDH1A1L3MBTL1
SCHEMBL3769333 0.68 KCNH2 (0.48) KCNH2MCHR1SLC2A1HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781650-A1 NOVEL COMPOUNDS HAVING AN ANTI-BACTERIAL ACTIVITY Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2007-05-09 EP disclosed
WO-2006021448-A1 NOVEL COMPOUNDS HAVING AN ANTI-BACTERIAL ACTIVITY Morphochem Aktiengesellschaft für kombinatorische Chemie (DE) 2006-03-02 WO disclosed