SCHEMBL5317581

SCHEMBL5317581

CC(=O)n1cc(CC(=O)O)c2cc([N+](=O)[O-])ccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.51
MAPT P10636 6/20 0.46
MEN1 O00255 5/20 0.46
KMT2A Q03164 5/20 0.46
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
NPSR1 Q6W5P4 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
HKDC1 Q2TB90 1/20 0.43
AKR1C3 P42330 4/20 0.43
AKR1C2 P52895 2/20 0.43
AKR1C4 P17516 1/20 0.43
PTGS1 P23219 1/20 0.43
PLA2G2A P14555 1/20 0.42
LMNA P02545 2/20 0.41
F2R P25116 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
F2RL3 Q96RI0 1/20 0.41
MTNR1A P48039 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28977334 0.79 AKR1C3 (0.65) AKR1C3AKR1C2AKR1C4PTGS1MTNR1A
SCHEMBL5320731 0.79 AKR1C3 (0.46) MAPTKDM4EALDH1A1AKR1C3AKR1C2
SCHEMBL28977349 0.79 AKR1C3 (0.58) MEN1KMT2AALDH1A1AKR1C3AKR1C2
SCHEMBL28977330 0.79 AKR1C3 (0.46) MAPTKDM4EALDH1A1AKR1C3AKR1C2
SCHEMBL6764463 0.76 KMT2A (0.49) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL8951254 0.76 PLA2G4A (0.71)
SCHEMBL31432746 0.75 CDC25A (0.55) MAPTKDM4EALDH1A1NPC1RAB9A
SCHEMBL8175848 0.73 CDK2 (0.46) CYP1A2MAPTMEN1KMT2AALDH1A1
SCHEMBL17871942 0.72 L3MBTL1 (0.52) MAPTMEN1KMT2AALDH1A1AKR1C3
SCHEMBL4229024 0.71 LCK (0.43) MEN1KMT2AALDH1A1NPSR1AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007075931-A2 REACTIVE HETEROCYCLIC DERIVATIVES AND METHODS FOR THEIR SYNTHESIS AND USE BIOSITE INCORPORATED (US) 2007-07-05 WO disclosed