SCHEMBL5317857

SCHEMBL5317857

CCOC(=O)c1ccc(C(F)(F)F)nc1C.CCOC(=O)c1ccc(C(F)(F)F)nc1C(F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.53
NPSR1 Q6W5P4 1/20 0.48
LMNA P02545 1/20 0.47
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
IDO1 P14902 1/20 0.46
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.44
TSHR P16473 2/20 0.44
CASP3 P42574 1/20 0.42
ATM Q13315 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
JUN P05412 2/20 0.42
NFKB1 P19838 2/20 0.42
NFKB2 Q00653 2/20 0.42
RELA Q04206 2/20 0.42
ALDH1A1 P00352 4/20 0.41
HPGD P15428 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5263472 0.95 KDM4E (0.49) KDM4ENPSR1LMNANPC1RAB9A
SCHEMBL4192553 0.94 KDM4E (0.58) KDM4ENPSR1LMNANPC1RAB9A
SCHEMBL31697314 0.93 KDM4E (0.50) KDM4ENPSR1LMNANPC1RAB9A
SCHEMBL1498542 0.93 KDM4E (0.50) KDM4ENPSR1LMNANPC1RAB9A
SCHEMBL6377043 0.81 KDM4E (0.59) KDM4ENPSR1IDO1MAPTTSHR
SCHEMBL3995268 0.81 KDM4E (0.53) KDM4ENPSR1LMNANPC1RAB9A
SCHEMBL24834467 0.80 KDM4E (0.48) KDM4ENPSR1IDO1MAPTTSHR
SCHEMBL29827383 0.80 KDM4E (0.48) KDM4ENPSR1NPC1RAB9AIDO1
SCHEMBL5077233 0.80 KDM4E (0.58) KDM4ENPSR1IDO1MAPTTSHR
SCHEMBL28944494 0.80 KDM4E (0.48) KDM4ENPSR1NPC1RAB9AIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1824828-A2 PYRIDINE BASED COMPOUNDS USEFUL AS INTERMEDIATES FOR PHARMACEUTICAL OR AGRICULTURAL END-PRODUCTS Peakdale Molecular Limited (GB) 2007-08-29 EP disclosed
WO-2006059103-A2 PYRIDINE BASED COMPOUNDS USEFUL AS INTERMEDIATES FOR PHARMACEUTICAL OR AGRICULTURAL END-PRODUCTS PEAKDALE MOLECULAR LIMITED (GB) 2006-06-08 WO disclosed