SCHEMBL5318236

SCHEMBL5318236

CCCN1CCCC(N(C)C(=O)c2ccc3c(c2)nc(N2CCOCC2)n3CCC)CC1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITK Q08881 16/20 0.49
CNR2 P34972 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
HRH3 Q9Y5N1 1/20 0.42
BCHE P06276 1/20 0.41
OPRM1 P35372 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5317398 0.91 ITK (0.49) ITKCNR2NPC1RAB9A
SCHEMBL5319079 0.88 ITK (0.49) ITKCNR2HRH3
SCHEMBL5316323 0.87 ITK (0.48) ITKCNR2HRH3
SCHEMBL5318216 0.83 ITK (0.43) ITKCNR2BCHEOPRM1
SCHEMBL5318430 0.80 ITK (0.49) ITKCNR2HRH3
SCHEMBL5318297 0.79 CNR2 (0.51) ITKCNR2
SCHEMBL5315733 0.78 PTGER4 (0.51)
SCHEMBL5319931 0.77 HRH3 (0.49) CNR2HRH3
SCHEMBL5315592 0.77 ITK (0.53) ITK
SCHEMBL5375164 0.75 KDM4E (0.54) CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007069053-A1 BENZIMIDAZOLE ANTAGONISTS OF THE H-3 RECEPTOR PFIZER PRODUCTS INC. (US) 2007-06-21 WO claimed
WO-2007069053-A1 BENZIMIDAZOLE ANTAGONISTS OF THE H-3 RECEPTOR PFIZER PRODUCTS INC. (US) 2007-06-21 WO disclosed