SCHEMBL5319947

SCHEMBL5319947

O=P(O)(O)C(F)(F)c1ccc(Cn2c3c(c4ccccc42)CCCC3)cc1Br

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.56
CA2 P00918 3/20 0.56
HDAC6 Q9UBN7 2/20 0.55
HDAC1 Q13547 1/20 0.55
HDAC10 Q969S8 1/20 0.55
HTR6 P50406 1/20 0.51
KDM4E B2RXH2 2/20 0.46
MEN1 O00255 1/20 0.46
GLA P06280 1/20 0.46
CASP1 P29466 1/20 0.46
CASP7 P55210 1/20 0.46
KMT2A Q03164 1/20 0.46
HSD17B10 Q99714 1/20 0.46
FABP4 P15090 3/20 0.46
ALDH1A1 P00352 1/20 0.45
PTPRC P08575 1/20 0.44
PTPN2 P17706 1/20 0.44
PTPN1 P18031 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5319152 0.99 CA1 (0.57) CA1CA2HDAC6HDAC1HDAC10
SCHEMBL5340406 0.99 CA1 (0.57) CA1CA2HDAC6HDAC1HDAC10
SCHEMBL14467239 0.99 CA1 (0.57) CA1CA2HDAC6HDAC1HDAC10
SCHEMBL5319783 0.88 PTGS1 (0.48) CA1CA2HDAC6HDAC1HDAC10
SCHEMBL5318871 0.88 PTGS1 (0.48) CA1CA2HDAC6HDAC1HDAC10
SCHEMBL5322648 0.86 PTPN1 (0.51) HDAC6HDAC1HDAC10KDM4EMEN1
SCHEMBL14467238 0.84 CA1 (0.59) CA1CA2HDAC6HDAC1HDAC10
SCHEMBL5344606 0.80 HDAC1 (0.53) HDAC6HDAC1HDAC10ALDH1A1PTPRC
SCHEMBL4106593 0.77 PTPN1 (0.49) HDAC6HDAC1KDM4EALDH1A1PTPRC
SCHEMBL5988010 0.77 PTPN1 (0.49) HDAC6HDAC1KDM4EALDH1A1PTPRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007081755-A2 INDOLE-BENZIMIDAZOLE AND INDAZOLE INHIBITORS OF TYROSINE PHOSPHATASES METABASIS THERAPEUTICS, INC. (US) 2007-07-19 WO disclosed