SCHEMBL5318871

SCHEMBL5318871

O=P(O)(O)C(F)(F)c1ccc(Cn2c3c(c4cc(Cl)ccc42)CCC3)cc1Br

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.48
PTGS2 P35354 1/20 0.48
CA1 P00915 3/20 0.45
CA2 P00918 3/20 0.45
HDAC6 Q9UBN7 3/20 0.44
HDAC1 Q13547 2/20 0.44
HDAC10 Q969S8 1/20 0.44
FABP4 P15090 1/20 0.40
LMNA P02545 3/20 0.40
HTT P42858 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
SLC2A1 P11166 1/20 0.40
HTR6 P50406 2/20 0.40
NR2F2 P24468 1/20 0.39
ACLY P53396 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5319783 0.99 PTGS1 (0.48) PTGS1PTGS2CA1CA2HDAC6
SCHEMBL5340406 0.89 CA1 (0.57) CA1CA2HDAC6HDAC1HDAC10
SCHEMBL5319947 0.88 CA1 (0.56) CA1CA2HDAC6HDAC1HDAC10
SCHEMBL14467239 0.87 CA1 (0.57) CA1CA2HDAC6HDAC1HDAC10
SCHEMBL5319152 0.87 CA1 (0.57) CA1CA2HDAC6HDAC1HDAC10
SCHEMBL5322648 0.75 PTPN1 (0.51) HDAC6HDAC1HDAC10SMN1; SMN2KDM4E
SCHEMBL7464584 0.75 CA1 (0.67) PTGS1PTGS2CA1CA2HDAC6
SCHEMBL14467238 0.75 CA1 (0.59) CA1CA2HDAC6HDAC1HDAC10
SCHEMBL4106593 0.73 PTPN1 (0.49) HDAC6HDAC1HTTKDM4EALDH1A1
SCHEMBL5988010 0.73 PTPN1 (0.49) HDAC6HDAC1HTTSMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007081755-A2 INDOLE-BENZIMIDAZOLE AND INDAZOLE INHIBITORS OF TYROSINE PHOSPHATASES METABASIS THERAPEUTICS, INC. (US) 2007-07-19 WO claimed
WO-2007081755-A2 INDOLE-BENZIMIDAZOLE AND INDAZOLE INHIBITORS OF TYROSINE PHOSPHATASES METABASIS THERAPEUTICS, INC. (US) 2007-07-19 WO disclosed