SCHEMBL5320893

SCHEMBL5320893

Cc1onc(NC(=O)OC(C)(C)C)c1F

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.35
CA2 P00918 1/20 0.35
CA12 O43570 1/20 0.34
CA9 Q16790 1/20 0.34
PSMB8 P28062 1/20 0.34
MLYCD O95822 1/20 0.33
HDAC3 O15379 2/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
CYP17A1 P05093 2/20 0.33
ATR Q13535 1/20 0.33
HDAC10 Q969S8 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
SYK P43405 1/20 0.32
LCK P06239 2/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3175510 0.84 CA1 (0.36) CA1CA2CA12CA9PSMB8
SCHEMBL16245702 0.83 CA1 (0.34) CA1CA2CA12CA9PSMB8
SCHEMBL24049964 0.81 KDM4E (0.49) CA1CA2CA12CA9PSMB8
SCHEMBL5347897 0.81 CA1 (0.36) CA1CA2CA12CA9PSMB8
SCHEMBL4411003 0.79 CA1 (0.36) CA1CA2CA12CA9PSMB8
SCHEMBL31319651 0.79 GABRA5 (0.36) CA1CA2CA12CA9PSMB8
SCHEMBL29953477 0.79 CA1 (0.33) CA1CA2CA12CA9PSMB8
SCHEMBL16245642 0.75 CA1 (0.35) CA1CA2CA12CA9PSMB8
SCHEMBL24049966 0.74 AAK1 (0.36) CA1CA2CA12CA9PSMB8
SCHEMBL27042890 0.73 CYP17A1 (0.34) CA1CA2CA12CA9PSMB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007109456-A2 SUBSTITUTED BIPHENYL ISOXAZOLE SULFONAMIDES AS DUAL ANGIOTENSIN ENDOTHELIN RECEPTOR ANTAGONISTS PHARMACOPEIA, INC. (US) 2007-09-27 WO disclosed