SCHEMBL5322971

SCHEMBL5322971

CN(C)c1ccc2c(c1)C(C1CCCCC1)=NN(Cc1ccccc1)C(=O)N2c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTH1R Q03431 14/20 0.54
APP P05067 1/20 0.39
MAPT P10636 1/20 0.39
SNCA P37840 1/20 0.39
CCKBR P32239 1/20 0.38
PTGS2 P35354 1/20 0.38
CASP1 P29466 1/20 0.38
CASP3 P42574 1/20 0.38
CASP4 P49662 1/20 0.38
CASP7 P55210 1/20 0.38
CASP9 P55211 1/20 0.38
CASP6 P55212 1/20 0.38
CASP8 Q14790 1/20 0.38
MCHR1 Q99705 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5321708 0.88 PTH1R (0.56) PTH1RCASP1CASP3CASP4CASP7
SCHEMBL5324664 0.88 PTH1R (0.58) PTH1RCCKBRCASP1CASP3CASP4
SCHEMBL5320334 0.87 PTH1R (0.69) PTH1RAPPMAPTSNCACCKBR
SCHEMBL5327910 0.85 PTH1R (0.56) PTH1RMAPTCCKBRMCHR1
SCHEMBL5325678 0.85 PTH1R (0.57) PTH1RCASP1CASP3CASP4CASP7
SCHEMBL5322753 0.84 PTH1R (0.61) PTH1RCCKBR
SCHEMBL5320657 0.83 PTH1R (0.64) PTH1RCCKBR
SCHEMBL5320380 0.80 PTH1R (0.57) PTH1RAPPMAPTSNCACCKBR
SCHEMBL5327453 0.79 PTH1R (0.45) PTH1RAPPMAPTSNCA
SCHEMBL5453686 0.79 PTH1R (0.47) PTH1RAPPMAPTSNCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129120-A9 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-03-22 WO disclosed
WO-2006129120-A2 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2006-12-07 WO disclosed