SCHEMBL5322980

SCHEMBL5322980

COc1cccc(C=C(Br)Br)c1O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR2 O60603 1/20 0.62
ERN1 O75460 1/20 0.62
TLR1 Q15399 1/20 0.62
TLR6 Q9Y2C9 1/20 0.62
CA12 O43570 1/20 0.56
POLB P06746 1/20 0.54
ADORA2A P29274 1/20 0.54
ADORA2B P29275 1/20 0.54
ADORA1 P30542 1/20 0.54
MAPT P10636 6/20 0.53
KDM4E B2RXH2 5/20 0.53
LMNA P02545 2/20 0.53
MAPK1 P28482 2/20 0.53
ALDH1A1 P00352 1/20 0.53
TP53 P04637 1/20 0.53
CYP3A4 P08684 1/20 0.53
HPGD P15428 1/20 0.53
ALOX15 P16050 1/20 0.53
ALOX12 P18054 1/20 0.53
HSD17B10 Q99714 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14198015 0.83 TLR2 (0.70) TLR2ERN1TLR1TLR6CA12
SCHEMBL10515793 0.82 NFE2L2 (0.52) CA12POLBMAPTKDM4ELMNA
SCHEMBL10401043 0.81 TLR2 (0.62) TLR2ERN1TLR1TLR6CA12
SCHEMBL5327152 0.80 TLR2 (0.43) TLR2ERN1TLR1TLR6CA12
SCHEMBL13457317 0.80 NFE2L2 (0.43) TLR2ERN1TLR1TLR6CA12
SCHEMBL4450612 0.79 ERN1 (0.96) TLR2ERN1TLR1TLR6CA12
SCHEMBL16004 0.77 ERN1 (1.00) TLR2ERN1TLR1TLR6CA12
SCHEMBL60623 0.77 TLR2 (0.67) TLR2ERN1TLR1TLR6CA12
SCHEMBL10054715 0.77 TLR2 (0.67) TLR2ERN1TLR1TLR6CA12
SCHEMBL11469615 0.77 TLR2 (0.67) TLR2ERN1TLR1TLR6CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007134421-A1 2-VINYL INDOLES, PYRIDO AND AZEPINO INDOLE DERIVATIVES, 2-ALKYNYL INDOLES, 2-ALKYNYL BENZO[b]FURANS, THEIR PRECURSORS AND NOVEL PROCESSES FOR THE PREPARATION THEREOF LAUTENS MARK (CA) 2007-11-29 WO disclosed
WO-2007134421-A1 2-VINYL INDOLES, PYRIDO AND AZEPINO INDOLE DERIVATIVES, 2-ALKYNYL INDOLES, 2-ALKYNYL BENZO[b]FURANS, THEIR PRECURSORS AND NOVEL PROCESSES FOR THE PREPARATION THEREOF LAUTENS MARK (CA) 2007-11-29 WO disclosed