SCHEMBL5323312

SCHEMBL5323312

NCc1c(-c2ccc(Cl)cc2Cl)ccc2c1CC(=O)[N]C2

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 19/20 0.43
DPP8 Q6V1X1 11/20 0.43
DPP9 Q86TI2 5/20 0.39
CYP3A4 P08684 4/20 0.39
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1996410 0.78 DPP4 (0.47) DPP4DPP8DPP9CYP3A4CYP2C19
SCHEMBL1997291 0.68 DPP4 (0.44) DPP4DPP8DPP9CYP3A4
SCHEMBL1995841 0.62 DPP4 (0.46) DPP4DPP8CYP3A4
SCHEMBL6224473 0.62 DPP4 (0.70) DPP4DPP8DPP9CYP3A4CYP2C19
SCHEMBL2000319 0.62 DPP4 (0.45) DPP4DPP8
SCHEMBL6221533 0.61 DPP4 (0.69) DPP4DPP8DPP9CYP3A4
SCHEMBL464507 0.61 AHR (0.64) CYP3A4
SCHEMBL29624840 0.61 AHR (0.64) CYP3A4
SCHEMBL8277153 0.61 DPP4 (0.64) DPP4DPP8CYP3A4
SCHEMBL3149261 0.61 DPP4 (1.00) DPP4DPP8CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007112347-A1 DIPEPTIDYL PEPTIDASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-10-04 WO claimed
WO-2007112347-A1 DIPEPTIDYL PEPTIDASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-10-04 WO disclosed