SCHEMBL5323913

SCHEMBL5323913

CC(C)[C@H](N)C(=O)N[C@H]([C]=O)Cc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSC P53634 7/20 0.55
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
CTRB1 P17538 3/20 0.48
CYP3A4 P08684 2/20 0.47
CYP1A2 P05177 1/20 0.47
CTSH P09668 1/20 0.47
CYP2D6 P10635 1/20 0.47
CTSK P43235 1/20 0.47
CTSL P07711 1/20 0.45
LMNA P02545 1/20 0.44
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8526731 0.90 CTSL (0.57) CTSKCTSL
SCHEMBL9143156 0.88 CTRB1 (0.61) CTSCNPC1RAB9ACTRB1CYP3A4
SCHEMBL27602044 0.88 CTRB1 (0.61) CTSCNPC1RAB9ACTRB1CYP3A4
SCHEMBL7316163 0.88 CTRB1 (0.61) CTSCNPC1RAB9ACTRB1CYP3A4
SCHEMBL7316156 0.88 CTRB1 (0.61) CTSCNPC1RAB9ACTRB1CYP3A4
SCHEMBL27788518 0.88 CTSC (0.57) CTSCNPC1RAB9ACTRB1CYP3A4
SCHEMBL9389290 0.84 CTSC (0.76) CTSCCYP3A4CYP1A2CTSHCYP2D6
SCHEMBL1691349 0.84 CTSC (0.76) CTSCCYP3A4CYP1A2CTSHCYP2D6
SCHEMBL583122 0.84 CTSC (0.76) CTSCCYP3A4CYP1A2CTSHCYP2D6
SCHEMBL583121 0.84 CTSC (0.76) CTSCCYP3A4CYP1A2CTSHCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106967062-A The analogs of novel C C 1065 and its conjugate 辛塔佳股份有限公司 2017-07-21 CN disclosed
CN-101415679-A Water-soluble CC-1065 analogs and conjugates thereof SINTAGAR B V (NL) 2009-04-22 CN disclosed
WO-2007112348-A2 PRODRUG COMPOSITION TSRL, INC. (US) 2007-10-04 WO disclosed
WO-1994018230-A1 INHIBITION OF HIV REPLICATION BY PEPTIDE-COPPER COMPLEXES PROCYTE CORPORATION (US) 1994-08-18 WO disclosed