SCHEMBL5324155

SCHEMBL5324155

NC1CCN(CCCF)CC1

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GNAI3 P08754 2/20 0.57
GNAO1 P09471 2/20 0.57
GNAI1 P63096 2/20 0.57
SPHK1 Q9NYA1 1/20 0.41
SIGMAR1 Q99720 3/20 0.41
HRH2 P25021 1/20 0.40
HRH1 P35367 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
KEAP1 Q14145 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ALOX15 P16050 1/20 0.35
HTR1D P28221 1/20 0.33
HTR1B P28222 1/20 0.33
OPRM1 P35372 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20618432 0.87 GNAI3 (0.44) GNAI3GNAO1GNAI1SPHK1SIGMAR1
SCHEMBL21584004 0.87 GNAI3 (0.44) GNAI3GNAO1GNAI1SPHK1SIGMAR1
SCHEMBL2803853 0.86 GNAI3 (0.50) GNAI3GNAO1GNAI1SPHK1HRH2
Hydrochloric Acid SCHEMBL2300838 0.84 GNAI3 (0.53) GNAI3GNAO1GNAI1SPHK1HRH2
Hydrochloric Acid SCHEMBL2293794 0.84 GNAI3 (0.53) GNAI3GNAO1GNAI1SPHK1HRH2
SCHEMBL3966764 0.84 GNAI3 (0.59) GNAI3GNAO1GNAI1SPHK1SIGMAR1
Hydrochloric Acid SCHEMBL3668361 0.82 GNAI3 (0.62) GNAI3GNAO1GNAI1SPHK1SIGMAR1
SCHEMBL23448772 0.79 GNAI3 (0.59) GNAI3GNAO1GNAI1SPHK1HRH2
SCHEMBL3973508 0.78 ALOX15 (0.60) GNAI3GNAO1GNAI1SPHK1SIGMAR1
SCHEMBL6889855 0.77 CARM1 (0.52) SIGMAR1HRH3OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116744920-A Heteroaryl piperidine derivative, and pharmaceutical composition and application thereof 贝达药业股份有限公司 2023-09-12 CN claimed
WO-2022166983-A1 HETEROARYLOPIPERIDINE DERIVATIVE, AND PHARMACEUTICAL COMPOSITION THEREOF AND USE THEREOF 贝达药业股份有限公司 2022-08-11 WO claimed
WO-2007134127-A2 AGENTS FOR IMAGING APOPTOSIS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2007-11-22 WO claimed
CN-116744920-A Heteroaryl piperidine derivative, and pharmaceutical composition and application thereof 贝达药业股份有限公司 2023-09-12 CN disclosed
WO-2022166983-A1 HETEROARYLOPIPERIDINE DERIVATIVE, AND PHARMACEUTICAL COMPOSITION THEREOF AND USE THEREOF 贝达药业股份有限公司 2022-08-11 WO disclosed
WO-2022166983-A1 HETEROARYLOPIPERIDINE DERIVATIVE, AND PHARMACEUTICAL COMPOSITION THEREOF AND USE THEREOF 贝达药业股份有限公司 2022-08-11 WO disclosed