SCHEMBL5324949

SCHEMBL5324949

Nc1ccc(N2C(=O)N(Cc3ccccc3)N=C(C3CCCCC3)c3cc(-c4cccnc4)ccc32)cc1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTH1R Q03431 12/20 0.57
BRD4 O60885 1/20 0.40
BACE1 P56817 2/20 0.39
CCR5 P51681 1/20 0.38
CYP11B2 P19099 2/20 0.38
CYP19A1 P11511 1/20 0.38
CYP11B1 P15538 1/20 0.38
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
WNT1 P04628 1/20 0.37
DYRK1A Q13627 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5320943 0.92 PTH1R (0.58) PTH1R
SCHEMBL5324210 0.89 PTH1R (0.59) PTH1R
SCHEMBL5323908 0.89 PTH1R (0.60) PTH1R
SCHEMBL5322494 0.86 PTH1R (0.56) PTH1R
SCHEMBL5329426 0.86 PTH1R (0.60) PTH1R
SCHEMBL5320402 0.85 PTH1R (0.62) PTH1R
SCHEMBL5280948 0.84 PTH1R (0.76) PTH1R
SCHEMBL5330994 0.81 PTH1R (0.43) PTH1RCYP11B2CYP19A1CYP11B1
SCHEMBL5324664 0.80 PTH1R (0.58) PTH1RBACE1
SCHEMBL5323705 0.79 PTH1R (0.79) PTH1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129120-A9 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-03-22 WO disclosed
WO-2006129120-A2 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2006-12-07 WO disclosed