SCHEMBL5325320

SCHEMBL5325320

CC1CN(c2c(Cl)cncc2Cl)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SUV39H2 Q9H5I1 2/20 0.49
GPR119 Q8TDV5 6/20 0.48
MAP4K4 O95819 1/20 0.48
HDAC1 Q13547 1/20 0.46
CYP3A4 P08684 1/20 0.41
SETD7 Q8WTS6 1/20 0.40
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
NTRK1 P04629 1/20 0.37
CCNC P24863 1/20 0.37
CDK8 P49336 1/20 0.37
NR1H2 P55055 2/20 0.37
GRM1 Q13255 1/20 0.36
SPR P35270 2/20 0.36
NR1H3 Q13133 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL38666762 0.82 MAP4K4 (0.53) SUV39H2GPR119MAP4K4HDAC1CYP3A4
SCHEMBL38665917 0.82 MAP4K4 (0.53) SUV39H2GPR119MAP4K4HDAC1CYP3A4
SCHEMBL29418786 0.81 GPR119 (0.48) SUV39H2GPR119MAP4K4HDAC1SETD7
SCHEMBL25214652 0.81 GPR119 (0.48) SUV39H2GPR119MAP4K4HDAC1SETD7
SCHEMBL16707804 0.80 GPR119 (0.42) SUV39H2GPR119CYP3A4ALDH1A1MAPT
SCHEMBL30045663 0.79 SUV39H2 (0.48) SUV39H2GPR119MAP4K4HDAC1SETD7
SCHEMBL23560874 0.79 MAP4K4 (0.54) SUV39H2GPR119MAP4K4HDAC1SETD7
SCHEMBL30005266 0.79 SUV39H2 (0.51) SUV39H2GPR119MAP4K4HDAC1NR1H2
SCHEMBL31173943 0.78 SUV39H2 (0.49) SUV39H2GPR119MAP4K4HDAC1NR1H2
SCHEMBL30419719 0.78 SUV39H2 (0.49) SUV39H2GPR119MAP4K4HDAC1NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007135427-A1 1,4-DISUBSTITUTED PIPERAZINE AND 1,4-DISUBSTITUTED AZEPANE AS 11 -BETA-HYDROXYSTEROID DEHYDROGENASE 1 INHIBITORS ASTRAZENECA AB (SE) 2007-11-29 WO disclosed