SCHEMBL532901

SCHEMBL532901

O=C(Oc1ccc(O)cc1)c1ccc(F)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.54
ATM Q13315 1/20 0.54
MEN1 O00255 2/20 0.54
HSD17B10 Q99714 1/20 0.50
SENP1 Q9P0U3 1/20 0.49
PARP10 Q53GL7 1/20 0.49
CA12 O43570 2/20 0.48
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
CA7 P43166 2/20 0.48
CA9 Q16790 2/20 0.48
CA14 Q9ULX7 2/20 0.48
MAPT P10636 1/20 0.48
F2 P00734 1/20 0.47
PRSS1 P07477 1/20 0.47
PRSS2 P07478 1/20 0.47
PRSS3 P35030 1/20 0.47
ELANE P08246 1/20 0.47
ESR1 P03372 1/20 0.46
ESR2 Q92731 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14640391 1.00 KMT2A (0.54) KMT2AATMMEN1HSD17B10SENP1
SCHEMBL14145708 1.00 KMT2A (0.54) KMT2AATMMEN1HSD17B10SENP1
SCHEMBL11311551 1.00 KMT2A (0.54) KMT2AATMMEN1HSD17B10SENP1
SCHEMBL14980966 0.95 SENP1 (0.53) KMT2AATMMEN1HSD17B10SENP1
SCHEMBL2838573 0.92 KMT2A (0.61) KMT2AATMMEN1HSD17B10PARP10
SCHEMBL29009176 0.92 KMT2A (0.61) KMT2AATMMEN1HSD17B10PARP10
SCHEMBL9696072 0.90 HSD17B10 (0.59) KMT2AMEN1HSD17B10SENP1PARP10
SCHEMBL740606 0.90 HSD17B10 (0.59) KMT2AMEN1HSD17B10SENP1PARP10
SCHEMBL688276 0.90 HSD17B10 (0.59) KMT2AMEN1HSD17B10SENP1PARP10
SCHEMBL16493489 0.90 HSD17B10 (0.59) KMT2AMEN1HSD17B10SENP1PARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 39 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1511713-B8 COMPOUNDS THAT ABROGATE DNA-DAMAGE-INDUCED CELL CYCLE G2 CHECKPOINT AND/OR AUGMENT THE ANTI-CANCER ACTIVITY OF DNA-DAMAGING TREATMENTS CANBAS CO LTD (JP) 2012-02-08 EP claimed
EP-1511713-B1 COMPOUNDS THAT ABROGATE DNA-DAMAGE-INDUCED CELL CYCLE G2 CHECKPOINT AND/OR AUGMENT THE ANTI-CANCER ACTIVITY OF DNA-DAMAGING TREATMENTS CANBAS CO LTD (JP) 2011-08-17 EP claimed
US-7652042-B2 Compounds that abrogate DNA damage induced cell cycle G2 checkpoint and/or augment anti-cancer activity of DNA-damaging treatments CANBAS CO., LTD. (JP) 2010-01-26 US claimed
CN-100577631-C The cell cycle G2 outpost of the tax office that the elimination dna damage causes and/or the compound that strengthens dna damage treatment antitumour activity CANBAS CO LTD 2010-01-06 CN claimed
US-7629364-B2 Compounds that abrogate DNA-damage-induced cell cycle G2 checkpoint and/or augment anti-cancer activity of DNA-damaging treatments CANBAS CO., LTD. (JP) 2009-12-08 US claimed
US-20080293137-A1 COMPOUNDS THAT ABROGATE DNA DAMAGE INDUCED CELL CYCLE G2 CHECKPOINT AND/OR AUGMENT ANTI-CANCER ACTIVITY OF DNA-DAMAGING TREATMENTS CANBAS CO., LTD. (JP) 2008-11-27 US claimed
US-20080227827-A1 COMPOUNDS THAT ABROGATE DNA DAMAGE INDUCED CELL CYCLE G2 CHECKPOINT AND/OR AUGMENT ANTI-CANCER ACTIVITY OF DNA-DAMAGING TREATMENTS CANBAS CO., LTD. (JP) 2008-09-18 US claimed
US-7407985-B2 Compounds that abrogate DNA damage induced cell cycle G2 checkpoint and/or augment anti-cancer activity of DNA-damaging treatments CANBAS CO., LTD. (JP) 2008-08-05 US claimed
JP-2007501608-A 2007-02-01 JP claimed
US-20060122269-A1 Compounds that abrogate DNA damage induced cell cycle G2 checkpoint and/or augment anti-cancer activity of DNA-damaging treatments CANBAS CO., LTD. (JP) 2006-06-08 US claimed
EP-1664340-A1 SENSITIVITY TEST TO PREDICT EFFICACY OF ANTI-CANCER THERAPIES Canbas Co., Ltd. (JP) 2006-06-07 EP claimed
US-7030111-B2 Compounds that abrogate DNA-damage-induced cell cycle G2 checkpoint and/or augment the anti-cancer activity of DNA damaging treatments CANBAS CO., LTD. (JP) 2006-04-18 US claimed
US-20060014157-A1 Sensitivity test to predict efficacy of anti-cancer therapies CANBAS CO., LTD. (JP) 2006-01-19 US claimed
CN-1671644-A Compounds that abrogate DNA-damage-induced cell cycle G2 checkpoint and/or augment the anti-cancer activity of DNA-damaging treatments CANBAS CO LTD (JP) 2005-09-21 CN claimed
EP-1511713-A2 COMPOUNDS THAT ABROGATE DNA-DAMAGE-INDUCED CELL CYCLE G2 CHECKPOINT AND/OR AUGMENT THE ANTI-CANCER ACTIVITY OF DNA-DAMAGING TREATMENTS Canbas Co. Ltd. (JP) 2005-03-09 EP claimed
WO-2005014856-A1 SENSITIVITY TEST TO PREDICT EFFICACY OF ANTI-CANCER THERAPIES CANBAS CO., LTD. (JP) 2005-02-17 WO claimed
US-20040198727-A1 Compounds that abrogate DNA-damage-induced cell cycle G2 checkpoint and/or augment the anti-cancer activity of DNA damaging treatments CANBAS CO., LTD. (JP) 2004-10-07 US claimed
WO-2003104181-A2 COMPOUNDS THAT ABROGATE DNA-DAMAGE-INDUCED CELL CYCLE G2 CHECKPOINT AND/OR AUGMENT THE ANTI-CANCER ACTIVITY OF DNA-DAMAGING TREATMENTS CANBAS CO. LTD. (JP) 2003-12-18 WO claimed
JP-58188838-A None JP disclosed
JP-S58188838-A ESTER DERIVATIVE OF 4-(4'-FLUOROBENZOYLOXY)PHENOL CHISSO CORP 1983-11-04 JP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080293137-A1 COMPOUNDS THAT ABROGATE DNA DAMAGE INDUCED CELL CYCLE G2 CHECKPOINT AND/OR AUGMENT ANTI-CANCER ACTIVITY OF DNA-DAMAGING TREATMENTS CDC25C, CHEK1, CDC25A KMT2A 883/4885ATM 128/4885MEN1 2545/4885
US-20040198727-A1 Compounds that abrogate DNA-damage-induced cell cycle G2 checkpoint and/or augment the anti-cancer activity of DNA damaging treatments CDC25C, CHEK1, DDB1 KMT2A 766/4885ATM 132/4885MEN1 2634/4885
US-20080227827-A1 COMPOUNDS THAT ABROGATE DNA DAMAGE INDUCED CELL CYCLE G2 CHECKPOINT AND/OR AUGMENT ANTI-CANCER ACTIVITY OF DNA-DAMAGING TREATMENTS CDC25C, CHEK1, CDC25A KMT2A 883/4885ATM 128/4885MEN1 2545/4885
US-20060122269-A1 Compounds that abrogate DNA damage induced cell cycle G2 checkpoint and/or augment anti-cancer activity of DNA-damaging treatments CDC25C, CHEK1, CDC25A KMT2A 883/4885ATM 128/4885MEN1 2545/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.