SCHEMBL533074

SCHEMBL533074

Cc1cc(C)c(NS(=O)(=O)c2cc(Cl)cc(Cl)c2O)c(C)c1NCC(C)(C)CN(C)C

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ACLY P53396 19/20 0.49
KMT2A Q03164 1/20 0.40
ACACB O00763 1/20 0.39
ACACA Q13085 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL534027 0.77 ACLY (0.55) ACLYACACBACACA
SCHEMBL533172 0.76 HSD17B2 (0.43) KMT2A
SCHEMBL532942 0.76 ACLY (0.51) ACLY
SCHEMBL533156 0.75 ACLY (0.56) ACLY
SCHEMBL533141 0.73 ACLY (0.63) ACLY
SCHEMBL532815 0.70 ACLY (0.53) ACLY
SCHEMBL533015 0.69 ACLY (0.54) ACLY
SCHEMBL14288686 0.69 ACLY (0.51) ACLYKMT2A
SCHEMBL8321880 0.68 ACLY (0.47) ACLY
SCHEMBL532884 0.68 ACLY (0.52) ACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2415760-A2 CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2012-02-08 EP disclosed
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed