SCHEMBL533138

SCHEMBL533138

Cc1cc(C)c(N2CCOCC2)c(C)c1NC(=O)c1ccccc1-c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
ALDH1A1 P00352 3/20 0.45
CHRNA7 P36544 2/20 0.45
CHRNA3 P32297 2/20 0.45
CHRNA4 P43681 2/20 0.45
LMNA P02545 1/20 0.45
CHRNA1 P02708 1/20 0.45
HTR3A P46098 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44
HSD17B10 Q99714 1/20 0.44
KDM4E B2RXH2 1/20 0.44
AVPR2 P30518 1/20 0.44
KMT2A Q03164 2/20 0.43
CNR2 P34972 1/20 0.43
MAPT P10636 1/20 0.43
TRPV4 Q9HBA0 1/20 0.43
CHRNB2 P17787 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL532826 0.90 ALDH1A1 (0.47) NPC1RAB9AALDH1A1CHRNA3CHRNA4
SCHEMBL532809 0.89 ALDH1A1 (0.46) NPC1RAB9AALDH1A1CHRNA3CHRNA4
SCHEMBL8320252 0.88 ALDH1A1 (0.46) RAB9AALDH1A1CHRNA3CHRNA4LMNA
SCHEMBL532902 0.84 L3MBTL1 (0.43) NPC1RAB9AALDH1A1CHRNA3CHRNA4
SCHEMBL533307 0.82 F10 (0.43) NPC1RAB9AALDH1A1LMNAL3MBTL1
SCHEMBL533536 0.82 L3MBTL1 (0.49) NPC1RAB9AALDH1A1LMNAL3MBTL1
SCHEMBL533668 0.82 HDAC7 (0.43) NPC1RAB9AALDH1A1CHRNA7CHRNA3
SCHEMBL532940 0.81 GAA (0.50) NPC1RAB9AALDH1A1LMNAL3MBTL1
SCHEMBL533116 0.80 MAPT (0.46) NPC1RAB9AALDH1A1LMNAL3MBTL1
SCHEMBL14288688 0.80 MTTP (0.52) ALDH1A1LMNAHPGDKDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2415760-A2 CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2012-02-08 EP disclosed
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed