SCHEMBL533142

SCHEMBL533142

ClC(Cl)c1cc[c]cc1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27524215 0.97 TSHR (0.48)
SCHEMBL533383 0.84 TSHR (0.42)
SCHEMBL7691395 0.77
SCHEMBL27674462 0.77
SCHEMBL22363110 0.77
SCHEMBL9529187 0.77
SCHEMBL11206282 0.77
SCHEMBL5075045 0.75 TSHR (0.67)
SCHEMBL3121541 0.75 LMNA (0.32)
SCHEMBL5249727 0.73 SLC6A2 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 193 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107022082-A A kind of application of silicon substrate hyperbranched conjugated polymer in Nitro-aromatic Compounds in Different detection 齐鲁工业大学 2017-08-08 CN claimed
CN-107022083-A A kind of silicon substrate hyperbranched conjugated polymer and preparation method thereof 齐鲁工业大学 2017-08-08 CN claimed
EP-2415763-B1 PHARMACEUTICAL COMPOSITION FOR TREATING OR PREVENTING GLAUCOMA UBE INDUSTRIES (JP) 2016-01-27 EP claimed
US-20140113907-A1 PYRIDYLAMINOACETIC ACID COMPOUND UBE INDUSTRIES, LTD. (JP) 2014-04-24 US claimed
EP-2520570-A1 AMINOPYRIDINE COMPOUND Ube Industries, Ltd. (JP) 2012-11-07 EP claimed
US-20120259123-A1 AMINOPYRIDINE COMPOUND UBE INDUSTRIES, LTD. (JP) 2012-10-11 US claimed
CN-102666490-A Aminopyridine compound UBE INDUSTRIES 2012-09-12 CN claimed
US-20120190852-A1 MEDICAL COMPOSITION FOR TREATMENT OR PROPHYLAXIS OF GLAUCOMA UBE INDUSTRIES, LTD. (JP) 2012-07-26 US claimed
CN-102448940-A Pharmaceutical composition for treating or preventing glaucoma UBE INDUSTRIES 2012-05-09 CN claimed
EP-2415763-A1 PHARMACEUTICAL COMPOSITION FOR TREATING OR PREVENTING GLAUCOMA Ube Industries, Ltd. (JP) 2012-02-08 EP claimed
US-20110054172-A1 PYRIDYLAMINOACETIC ACID COMPOUND UBE CORPORATION (JP) 2011-03-03 US claimed
CN-101970410-A Pyridylaminoacetic acid compounds UBE INDUSTRIES 2011-02-09 CN claimed
EP-2264009-A1 PYRIDYLAMINOACETIC ACID COMPOUND Ube Industries, Ltd. (JP) 2010-12-22 EP claimed
EP-1653960-A4 MELANIN CONCENTRATING HORMONE RECEPTOR ANTAGONIST AMGEN INC (US) 2008-11-26 EP claimed
EP-1899339-A1 1,2-DIHYDRO-SPIRO(3H-INDOLE-3-4 -PIPERIDINE) COMPOUNDS AS MODULATORS OF THE MAS RECEPTOR NOVEL Arena Pharmaceuticals, Inc. (US) 2008-03-19 EP claimed
WO-2007002114-A1 1,2-DIHYDRO-SPIRO(3H-INDOLE-3-4’-PIPERIDINE) COMPOUNDS AS MODULATORS OF THE MAS RECEPTOR NOVEL ARENA PHARMACEUTICALS, INC. (US) 2007-01-04 WO claimed
EP-1653960-A2 MELANIN CONCENTRATING HORMONE RECEPTOR ANTAGONIST AMGEN INC. (US) 2006-05-10 EP claimed
US-20050215526-A1 Melanin concentrating hormone receptor antagonist AMGEN, INC. 2005-09-29 US claimed
WO-2005019167-A2 MELANIN CONCENTRATING HORMONE RECEPTOR ANTAGONIST AMGEN, INC. (US) 2005-03-03 WO claimed
WO-2024151706-A1 FUNCTIONALIZATION OF SOLUBLE POLYDIENES AND POLYISOPRENES USING DITHIOPHOSPHORIC ACIDS ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2024-07-18 WO disclosed
US-20240194920-A1 CARBENIUM BASED ORGANIC REDOX FLOW BATTERIES ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2024-06-13 US disclosed
US-20240085753-A1 ELECTROCHROMIC COMPOSITION AND ELECTROCHROMIC DEVICE TAI YING OPTRONICS CO., LTD. (TW) 2024-03-14 US disclosed
US-11769905-B2 Poly(alkylene oxide) siloxane-based electrolytes for rechargeable batteries UCHICAGO ARGONNE, LLC (US) 2023-09-26 US disclosed
WO-2023164025-A1 REGENERATION OF SYMMETRICAL NONAQUEOUS ORGANIC REDOX FLOW BATTERIES ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2023-08-31 WO disclosed
EP-4178576-A1 DEOXYNOJIRIMYCIN DERIVATIVES AS GLUCOSIDASE INHIBITORS Emergent Product Development Gaithersburg Inc. (US) 2023-05-17 EP disclosed
EP-4139981-A1 CARBENIUM BASED ORGANIC REDOX FLOW BATTERIES Arizona Board of Regents on behalf of The University of Arizona (US) 2023-03-01 EP disclosed
CN-115298164-A Process for preparing 4-cyanobenzoyl chlorides 巴斯夫欧洲公司 2022-11-04 CN disclosed
WO-2022011211-A1 DEOXYNOJIRIMYCIN DERIVATIVES AS GLUCOSIDASE INHIBITORS EMERGENT PRODUCT DEVELOPMENT GAITHERSBURG INC. (US) 2022-01-13 WO disclosed
WO-2021217092-A1 CARBENIUM BASED ORGANIC REDOX FLOW BATTERIES ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2021-10-28 WO disclosed
EP-3215499-B1 IMINOSUGARS USEFUL FOR THE TREATMENT OF VIRAL DISEASES EMERGENT VIROLOGY LLC (US) 2021-01-20 EP disclosed
US-20200384115-A1 TARGETED DELIVERY TO BETA CELLS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2020-12-10 US disclosed
US-10840531-B2 Two-electron redox active molecules with high capacity and energy density for energy storage applications UCHICAGO ARGONNE, LLC (US) 2020-11-17 US disclosed
EP-3612232-A1 TARGETED DELIVERY TO BETA CELLS The Broad Institute, Inc. (US) 2020-02-26 EP disclosed
US-10428022-B2 Iminosugars useful for the treatment of viral diseases EMERGENT VIROLOGY LLC (US) 2019-10-01 US disclosed
US-20190051921-A1 TWO-ELECTRON REDOX CATHOLYTE FOR REDOX FLOW BATTERIES UCHICAGO ARGONNE, LLC 2019-02-14 US disclosed
US-20190044181-A1 POLY(ALKYLENE OXIDE) SILOXANE-BASED ELECTROLYTES FOR RECHARGEABLE BATTERIES UNITED STATES DEPARTMENT OF ENERGY 2019-02-07 US disclosed
US-20180354991-A1 THERAPEUTIC COMPOSITIONS INCLUDING GRAMICIDIN S PEPTIDYL CONJUGATES OR IMIDAZOLE-SUBSTITUTED FATTY ACIDS, VARIANTS THEREOF AND USES THEREOF STEALTH PEPTIDES INTERNATIONAL, INC. (MC) 2018-12-13 US disclosed
WO-2018195486-A1 TARGETED DELIVERY TO BETA CELLS THE BROAD INSTITUTE, INC. (US) 2018-10-25 WO disclosed
US-20180273473-A1 IMINOSUGARS USEFUL FOR THE TREATMENT OF VIRAL DISEASES EMERGENT PRODUCT DEVELOPMENT GAITHERSBURG INC. 2018-09-27 US disclosed
CN-108431092-A The continuation method reacted with particle alkali metal dispersion CHT R.拜特利希有限公司 2018-08-21 CN disclosed
US-10026984-B2 Multi-electron redox active molecules for energy storage applications UCHICAGO ARGONNE, LLC (US) 2018-07-17 US disclosed
CN-105777482-B A kind of 1-(1- chloromethyl vinyl bases)The synthetic method of -2,4- difluorobenzene 浙江大学宁波理工学院 2018-06-15 CN disclosed
US-9991542-B2 Two-electron high potential and high capacity redox active molecules for energy storage applications UCHICAGO ARGONNE, LLC (US) 2018-06-05 US disclosed
US-20180042983-A1 THERAPEUTIC COMPOSITIONS INCLUDING MITOCHONDRIAL FISSION INHIBITOR PEPTIDES, VARIANTS THEREOF, AND METHODS OF USING THE SAME STEALTH PEPTIDES INTERNATIONAL, INC. (MC) 2018-02-15 US disclosed
EP-3256143-A2 THERAPEUTIC COMPOSITIONS INCLUDING MITOCHONDRIAL FISSION INHIBITOR PEPTIDES, VARIANTS THEREOF AND METHODS OF USING THE SAME Stealth Peptides International, Inc. (MC) 2017-12-20 EP disclosed
EP-3215499-A1 IMINOSUGARS USEFUL FOR THE TREATMENT OF VIRAL DISEASES Emergent Virology LLC (US) 2017-09-13 EP disclosed
CN-107022082-A A kind of application of silicon substrate hyperbranched conjugated polymer in Nitro-aromatic Compounds in Different detection 齐鲁工业大学 2017-08-08 CN disclosed
CN-107022083-A A kind of silicon substrate hyperbranched conjugated polymer and preparation method thereof 齐鲁工业大学 2017-08-08 CN disclosed
CN-106967076-A One kind has 6H dibenzopyrans structural compounds and preparation method thereof 河南师范大学 2017-07-21 CN disclosed
CN-104327200-B The preparation method of polyalphaolefin 埃克森美孚化学专利公司 2017-07-14 CN disclosed
CN-104211967-B Polymetalcarbosilane, and preparation method and application thereof 中国科学院过程工程研究所 2017-05-03 CN disclosed
US-20170062842-A1 TWO-ELECTRON REDOX ACTIVE MOLECULES WITH HIGH CAPACITY AND ENERGY DENSITY FOR ENERGY STORAGE APPLICATIONS UCHICAGO ARGONNE, LLC 2017-03-02 US disclosed
US-20170062863-A1 TWO-ELECTRON HIGH POTENTIAL AND HIGH CAPACITY REDOX ACTIVE MOLECULES FOR ENERGY STORAGE APPLICATIONS UCHICAGO ARGONNE, LLC 2017-03-02 US disclosed
US-20170062862-A1 MULTI-ELECTRON REDOX ACTIVE MOLECULES FOR ENERGY STORAGE APPLICATIONS UCHICAGO ARGONNE, LLC 2017-03-02 US disclosed
WO-2016209261-A1 THERAPEUTIC COMPOSITIONS INCLUDING GRAMICIDIN S PEPTIDYL CONJUGATES OR IMIDAZOLE-SUBSTITUTED FATTY ACIDS, VARIANTS THEREOF, AND USES THEREOF STEALTH BIOTHERAPEUTICS CORP (MC) 2016-12-29 WO disclosed
WO-2016200364-A1 THERAPEUTIC COMPOSITIONS INCLUDING SkQ COMPOUNDS AND USES THEREOF STEALTH PEPTIDES INTERNATIONAL, INC. (MC) 2016-12-15 WO disclosed
WO-2016195663-A1 THERAPEUTIC COMPOSITIONS INCLUDING BPM 31510, VARIANTS AND ANALOGUES THEREOF, AND USES THEREOF STEALTH PEPTIDES INTERNATIONAL, INC. (MC) 2016-12-08 WO disclosed
WO-2016190852-A1 THERAPEUTIC COMPOSITIONS INCLUDING CHROMANYL COMPOUNDS, VARIANTS AND ANALOGUES THEREOF, AND USES THEREOF STEALTH PEPTIDES INTERNATIONAL, INC. (MC) 2016-12-01 WO disclosed
WO-2016130143-A2 THERAPEUTIC COMPOSITIONS INCLUDING MITOCHONDRIAL FISSION INHIBITOR PEPTIDES, VARIANTS THEREOF AND METHODS OF USING THE SAME STEALTH PEPTIDES INTERNATIONAL, INC. (MC) 2016-08-18 WO disclosed
CN-105829294-A METHYLENE LINKED QUINOLINYL MODULATORS OF ROR-GAMMA-T 詹森药业有限公司 2016-08-03 CN disclosed
WO-2016073652-A1 IMINOSUGARS USEFUL FOR THE TREATMENT OF VIRAL DISEASES UNITHER VIROLOGY, LLC (US) 2016-05-12 WO disclosed
EP-2415763-B1 PHARMACEUTICAL COMPOSITION FOR TREATING OR PREVENTING GLAUCOMA UBE INDUSTRIES (JP) 2016-01-27 EP disclosed
WO-2016004093-A2 THERAPEUTIC COMPOSITIONS INCLUDING GALECTIN-3 INHIBITORS AND USES THEREOF STEALTH BIOTHERAPEUTICS CORP (MC) 2016-01-07 WO disclosed
CN-102781884-B Process for producing alpha-olefin oligomer MITSUBISHI CHEMICAL CORP. (JP) 2015-11-25 CN disclosed
CN-102448940-B For the medical composition of glaucomatous treatment or prevention UBE INDUSTRIES, LTD. (JP) 2015-10-21 CN disclosed
CN-104926589-A Process for producing alpha-olefin oligomer MITSUBISHI CHEM CORP 2015-09-23 CN disclosed
CN-103965099-A Pyridylaminoacetic Acid Compound UBE INDUSTRIES 2014-08-06 CN disclosed
CN-101970410-B Pyridylaminoacetic acid compounds UBE INDUSTRIES 2014-06-25 CN disclosed
US-20140113907-A1 PYRIDYLAMINOACETIC ACID COMPOUND UBE INDUSTRIES, LTD. (JP) 2014-04-24 US disclosed
US-8648097-B2 Pyridylaminoacetic acid compound UBE INDUSTRIES, LTD. (JP) 2014-02-11 US disclosed
CN-102781884-A Process for producing alpha-olefin oligomer MITSUBISHI CHEM CORP 2012-11-14 CN disclosed
EP-2520570-A1 AMINOPYRIDINE COMPOUND Ube Industries, Ltd. (JP) 2012-11-07 EP disclosed
US-20120259123-A1 AMINOPYRIDINE COMPOUND UBE INDUSTRIES, LTD. (JP) 2012-10-11 US disclosed
CN-102666490-A Aminopyridine compound UBE INDUSTRIES 2012-09-12 CN disclosed
US-20120190852-A1 MEDICAL COMPOSITION FOR TREATMENT OR PROPHYLAXIS OF GLAUCOMA UBE INDUSTRIES, LTD. (JP) 2012-07-26 US disclosed
CN-102448940-A Pharmaceutical composition for treating or preventing glaucoma UBE INDUSTRIES 2012-05-09 CN disclosed
US-8114886-B2 Pyridylmethylsulfone derivative DAIICHI SANKYO COMPANY, LIMITED (JP) 2012-02-14 US disclosed
EP-2415763-A1 PHARMACEUTICAL COMPOSITION FOR TREATING OR PREVENTING GLAUCOMA Ube Industries, Ltd. (JP) 2012-02-08 EP disclosed
CN-101107260-B Transition metal complex, method for producing the same, substituted fluorene compound, method for producing the substituted fluorene compound, catalyst component for olefin polymerization, catalyst for olefin polymerization, and method for producing olefin polymer SUMITOMO CHEMICAL CO.,LTD. (JP) 2012-02-08 CN disclosed
CN-101163678-B Pyridylmethylsulfone derivative DAIICHI SANKYO CO LTD 2012-01-04 CN disclosed
US-20110054172-A1 PYRIDYLAMINOACETIC ACID COMPOUND UBE CORPORATION (JP) 2011-03-03 US disclosed
CN-101970410-A Pyridylaminoacetic acid compounds UBE INDUSTRIES 2011-02-09 CN disclosed
EP-2264009-A1 PYRIDYLAMINOACETIC ACID COMPOUND Ube Industries, Ltd. (JP) 2010-12-22 EP disclosed
US-20100222330-A1 New Compounds BIOVITRUM AB (SE) 2010-09-02 US disclosed
US-7659276-B2 Melanin concentrating hormone receptor antagonist AMGEN, INC. (US) 2010-02-09 US disclosed
CN-100584462-C Bimetallic catalyst with high activity EXXONMOBIL CHEMICAL PATENT CO 2010-01-27 CN disclosed
US-7572787-B2 Substituted naphthalene sulfonamides BIOVITRUM AB (SE) 2009-08-11 US disclosed
US-20090149439-A1 PYRIDYLMETHYSULFONE DERIVATIVE DAIICHI SANKYO COMPANY LIMITED (JP) 2009-06-11 US disclosed
US-20090143405-A1 MELANIN CONCENTRATING HORMONE RECEPTOR ANTAGONIST AMGEN, INC. (US) 2009-06-04 US disclosed
CN-101402601-A Substituted sulfonamide compounds, process for their use as medicament for the treatment of cns disorders, obesity and type ii diabetes BIOVITRUM AB PUBL (SE) 2009-04-08 CN disclosed
US-7514438-B2 Melanin concentrating hormone receptor antagonist AMGEN, INC. (US) 2009-04-07 US disclosed
CN-100457726-C Substituted sulfonamide compounds, process for their preparation and their use as medicaments for the treatment of CNS disorders, obesity and type II diabetes CAMBRIDGE BIOTECHNOLOGY LTD (SE) 2009-02-04 CN disclosed
EP-1653960-A4 MELANIN CONCENTRATING HORMONE RECEPTOR ANTAGONIST AMGEN INC (US) 2008-11-26 EP disclosed
EP-1675830-A4 HETEROCYCLIC AMIDES AND SULFONAMIDES SCIOS INC (US) 2008-08-20 EP disclosed
CN-101163678-A Pyridylmethylsulfone derivative DAIICHI SANKYO CO LTD (JP) 2008-04-16 CN disclosed
CN-100371351-C Organometal catalyst compositions PHILLIPS PETROLEUM CO (US) 2008-02-27 CN disclosed
CN-101107260-A Transition metal complex, method for producing the same, substituted fluorene compound, method for producing the substituted fluorene compound, catalyst component for olefin polymerization, catalyst for olefin polymerization, and method for producing olefin polymer SUMITOMO CHEMICAL CO (JP) 2008-01-16 CN disclosed
EP-1867636-A1 PYRIDYLMETHYLSULFONE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2007-12-19 EP disclosed
CN-101062959-A Method of making mixed ziegler-natta/metallocece catalysts EXXONMOBIL CHEM PATENTS INC (US) 2007-10-31 CN disclosed
US-7276511-B2 Benzylamine derivative ZERIA PHARMACEUTICAL CO., LTD. (JP) 2007-10-02 US disclosed
CN-1319995-C Reactor wall coating and method of forming the same UNIVATION TECH LLC (US) 2007-06-06 CN disclosed
US-20070066598-A1 Compounds BIOVITRUM AB, A SWEDEN CORPORATION 2007-03-22 US disclosed
US-20070066599-A1 New compounds BIOVITRUM AB, A SWEDEN CORPORATION 2007-03-22 US disclosed
US-20070066600-A1 Compounds PROXIMAGEN NEUROSCIENCE PLC (GB) 2007-03-22 US disclosed
CN-1301190-C Laminated film JAPAN POLYCHEM CORP (JP) 2007-02-21 CN disclosed
US-7144883-B2 Bicyclic sulfonamide compounds BIOVITRUM AB (SE) 2006-12-05 US disclosed
CN-1868583-A Organometal catalyst compositions PHILLIPS PETROLEUM CO (US) 2006-11-29 CN disclosed
US-20060199821-A1 Heterocyclic amides and sulfonamides SCIOS, INC. (US) 2006-09-07 US disclosed
CN-1829689-A Phenylmethylamine derivatives ZERIA PHARM CO LTD (JP) 2006-09-06 CN disclosed
US-20060194841-A1 E.g., N-{2-(3,4-dichlorophenyl)-2-[(3,3-diphenylpropionyl)-methylamino]-4-{spiro[benzo(c)thiophene-1(3H),4'-piperidine]-(2S)-oxide}-1'-yl-butyl}-3,3,3-trifluoro-N-methyl-propionamide hydrochloride, NK-1 or NK-2 receptor antagonists; irritable bowel syndrome, pain, anxiety, COPD, headaches and vomiting ZERIA PHARMACEUTICAL CO., LTD. (JP) 2006-08-31 US disclosed
CN-1267191-C organometallic catalyst composition PHILLIPS PETROLEUM CO (US) 2006-08-02 CN disclosed
US-7084137-B2 Thiazines and thiazoles as agents for protecting materials BAYER AKTIENGESELLSCHAFT (DE) 2006-08-01 US disclosed
CN-1800185-A Substituted sulfonamide compounds, process for their use as medicament for the treatment of CNS disorders, obesity and type II diabetes. BIOVITRUM AB (SE) 2006-07-12 CN disclosed
EP-1675830-A2 HETEROCYCLIC AMIDES AND SULFONAMIDES SCIOS INC. (US) 2006-07-05 EP disclosed
EP-1653960-A2 MELANIN CONCENTRATING HORMONE RECEPTOR ANTAGONIST AMGEN INC. (US) 2006-05-10 EP disclosed
EP-1650189-A1 BENZYLAMINE DERIVATIVE Zeria Pharmaceutical Co., Ltd. (JP) 2006-04-26 EP disclosed
CN-1231294-C Organic metal catalyst composition PHILLIPS PETROLEUM CO (US) 2005-12-14 CN disclosed
CN-1691979-A Bimetallic catalysts with higher activity EXXONMOBIL CHEM PATENTS INC (US) 2005-11-02 CN disclosed
CN-1688608-A Reactor wall coating and processes for forming same UNIVATION TECH LLC (US) 2005-10-26 CN disclosed
US-20050215526-A1 Melanin concentrating hormone receptor antagonist AMGEN, INC. 2005-09-29 US disclosed
CN-1625440-A Bimetallic catalyst with high activity EXXONMOBIL CHEMICAL PATENT CO (US) 2005-06-08 CN disclosed
CN-1202138-C Organometal catalyst compositions PHILLIPS PETROLEUM CO (US) 2005-05-18 CN disclosed
WO-2005033072-A2 HETEROCYCLIC AMIDES AND SULFONAMIDES SCIOS INC. (US) 2005-04-14 WO disclosed
WO-2005019167-A2 MELANIN CONCENTRATING HORMONE RECEPTOR ANTAGONIST AMGEN, INC. (US) 2005-03-03 WO disclosed
CN-1188431-C Organometal compound catalyst PHILLIPS PETROLEUM CO (US) 2005-02-09 CN disclosed
CN-1558826-A Laminated film 日本聚丙烯公司 2004-12-29 CN disclosed
US-20040204405-A1 Thiazines and thiazoles as agents for protecting materials LANXESS DEUTSCHLAND GMBH (DE) 2004-10-14 US disclosed
CN-1522245-A Substituted sulfonamide compounds, process for their preparation and their use as medicaments for the treatment of CNS disorders, obesity and type II diabetes �Ȱ�ά����ķ�ɷݹ�˾ 2004-08-18 CN disclosed
EP-1437940-A1 THIAZINES AND THIAZOLES FOR USE AS MATERIAL PROTECTIVE AGENTS Bayer Chemicals AG (DE) 2004-07-21 EP disclosed
EP-1412325-A1 SUBSTITUTED SULFONAMIDE COMPOUNDS, PROCESS FOR THEIR USE AS MEDICAMENT FOR THE TREATMENT OF CNS DISORDERS, OBESITY AND TYPE II DIABETES BIOVITRUM AB (SE) 2004-04-28 EP disclosed
CN-1137902-C Supported polymerization catalysts 2004-02-11 CN disclosed
CN-1128168-C Process for preparing polyolefin compositions MITSUI CHEMICALS INC (JP) 2003-11-19 CN disclosed
US-20030158202-A1 Substituted fused ring sulfonamides containing, e.g., naphthalene, isoquinoline, quinoline, benzofuran or benzothiophene rings; treatment of conditions relating to obesity, type II diabetes and CNS disorders PROXIMAGEN NEUROSCIENCE PLC (GB) 2003-08-21 US disclosed
US-20030129081-A1 Thiazines and thiazoles as agents for protecting materials BAYER AKTIENGESELLSCHAFT (DE) 2003-07-10 US disclosed
CN-1110366-C Non-pyrophoric solids BASF AG (DE) 2003-06-04 CN disclosed
CN-1414978-A Organometal catalyst compositions PHILLIPS PETROLEUM CO (US) 2003-04-30 CN disclosed
CN-1414880-A Organometal compound catalyst PHILLIPS PETROLEUM CO (US) 2003-04-30 CN disclosed
CN-1404491-A Process for producing polyolefin composition MITSUI CHEMICALS INC (JP) 2003-03-19 CN disclosed
WO-2003001913-A1 THIAZINES AND THIAZOLES FOR USE AS MATERIAL PROTECTIVE AGENTS BAYER CHEMICALS AG (DE) 2003-01-09 WO disclosed
WO-2002100822-A1 SUBSTITUTED SULFONAMIDE COMPOUNDS, PROCESS FOR THEIR USE AS MEDICAMENT FOR THE TREATMENT OF CNS DISORDERS, OBESITY AND TYPE II DIABETES BIOVITRUM AB (SE) 2002-12-19 WO disclosed
CN-1377373-A organometallic catalyst composition PHILLIPS PETROLEUM CO (US) 2002-10-30 CN disclosed
CN-1376167-A organometallic catalyst composition PHILLIOPS PETROLEUM COMPANY (US) 2002-10-23 CN disclosed
CN-1092659-C Novel pyrimidine derivative OTSUKA PHARMA CO LTD (JP) 2002-10-16 CN disclosed
CN-1373373-A Oblique raster type light isolator and its preparing process HAO MING (CN) 2002-10-09 CN disclosed
CN-1323319-A Supported polymerization catalysts BOREALIS AS (FI) 2001-11-21 CN disclosed
CN-1070487-C Hexahydronaphthalene ester derivatives, their preparation and their therapeutic uses SANKYO CO (JP) 2001-09-05 CN disclosed
CN-1304800-A Organic metal catalyst composition PHILLIPS PETROLEUM CO (US) 2001-07-25 CN disclosed
CN-1301600-A organometallic catalyst composition PHILLIPS PETROLEUM CO (US) 2001-07-04 CN disclosed
US-6242449-B1 TREATING PROSTATIC HYPERTROPHY, URINATION DISORDERS ASSOCIATED WITH PROSTATIC HYPERTROPHY, MALE PATTERN ALOPECIA, OR ACNE ZERIA PHARMACEUTICAL CO., LTD. (JP) 2001-06-05 US disclosed
CN-1292007-A Method for making polymer blends by using series reactors EXXON CHEMICAL PATENTS INC (US) 2001-04-18 CN disclosed
US-6197774-B1 THERAPY FOR ASTHMA, SKIN DISORDERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2001-03-06 US disclosed
CN-1264365-A 3-benzoylindole derivatives and drugs containing the same ZERIA PHARM CO LTD (JP) 2000-08-23 CN disclosed
EP-1019501-A1 NOVEL PYRIMIDINE DERIVATIVE OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2000-07-19 EP disclosed
CN-1052734-C Propylene elastomer MITSUI PETROCHEMICAL IND (JP) 2000-05-24 CN disclosed
EP-0997457-A1 3-BENZOYLINDOLE DERIVATIVES AND DRUGS CONTAINING THE SAME ZERIA PHARMACEUTICAL CO., LTD. (JP) 2000-05-03 EP disclosed
CN-1251057-A Non self-igniting solid BASF AG (DE) 2000-04-19 CN disclosed
CN-1250450-A Novel pyrimidine derivative OTSUKA PHARMA CO LTD (JP) 2000-04-12 CN disclosed
CN-1048733-C Prepolymerized catalyst, catalyst for olefin polymerization, polymerization process of olefin, and olefin polymer MITSUI PETROCHEMICAL IND (JP) 2000-01-26 CN disclosed
CN-1043144-C Prepolymerized catalyst, catalyst for olefin polymerization, and process for olefin polymerization MITSUI CHEMICALS INC (JP) 1999-04-28 CN disclosed
EP-0765351-B1 AMIDATION OF ESTER FUNCTIONALIZED HYDROCARBON POLYMERS EXXON CHEMICAL PATENTS INC (US) 1999-01-13 EP disclosed
WO-1998041526-A1 NOVEL PYRIMIDINE DERIVATIVE OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-09-24 WO disclosed
US-5627259-A REACTION OF OLEFIN POLYMERS WITH CARBON MONOXIDE AND ALCOHOL THEN REACTION OF ESTER WITH POLYAMINE COMPOUND RELEASING ALCOHOL COMPOUND EXXON CHEMICAL PATENTS INC. (US) 1997-05-06 US disclosed
EP-0765351-A1 AMIDATION OF ESTER FUNCTIONALIZED HYDROCARBON POLYMERS EXXON CHEMICAL PATENTS INC. (US) 1997-04-02 EP disclosed
WO-1995035330-A1 AMIDATION OF ESTER FUNCTIONALIZED HYDROCARBON POLYMERS EXXON CHEMICAL PATENTS INC. (US) 1995-12-28 WO disclosed
CN-1113494-A Prepolymerized catalyst, catalyst for olefin polymerization, polymerization process of olefin, and olefin polymer MITSUI PETROCHEMICAL IND (JP) 1995-12-20 CN disclosed
CN-1029405-C Lipid A analogs having immunoactivating and anti-tumor activity SANKYO CO (JP) 1995-08-02 CN disclosed
EP-0282895-B1 2-oxa-isocephem compounds, compositions containing same and processes for preparing same OTSUKA PHARMA CO LTD (JP) 1995-06-07 EP disclosed
CN-1091432-A Can suppress the active peptide of hiv protease, its preparation with and medical use SANKYO CO (JP) 1994-08-31 CN disclosed
CN-1091128-A Piperidine derivative SANKYO CO (JP) 1994-08-24 CN disclosed
CN-1023801-C 2-Oxa-isocephem compounds, compositions containing same and processes for preparing same OTSUKA PHARMA CO LTD (JP) 1994-02-16 CN disclosed
CN-1070651-A Catalyst for olefin polymerization and olefin polymer MITSUI PETROCHEMICAL IND (JP) 1993-04-07 CN disclosed
EP-0320733-B1 2-TERT.-BUTYL-5-ISOXAZOLYL METHYLTHIO-3(2H)-PYRIDAZIN-3-ONE DERIVATIVES BASF Aktiengesellschaft (DE) 1993-03-03 EP disclosed
US-5126461-A Silica in organic solution SHELL RESEARCH LIMITED (GB) 1992-06-30 US disclosed
US-5037976-A Antimicrobial Agent OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-08-06 US disclosed
EP-0437016-A2 Lipid A analogues having immunoactivating and anti-tumour activity Sankyo Company Limited (JP) 1991-07-17 EP disclosed
EP-0243173-B1 NEW DIPHOSPHONIC ACID COMPOUNDS, PROCESSES FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-06-26 EP disclosed
CN-1052481-A Lipoid category-A with immunocompetence and anti-tumor activity is like thing SANKYO CO (JP) 1991-06-26 CN disclosed
EP-0432818-A2 Process for opening cyclopropane rings SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1991-06-19 EP disclosed
US-4963530-A Renin inhibitor peptide compounds, a process for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL COMPANY, LTD. (JP) 1990-10-16 US disclosed
US-4963536-A INHIBIT BONE RESORPTION FUJISAWA PHARMACEUTICAL COMPANY, LTD. (JP) 1990-10-16 US disclosed
US-4929617-A INSECTICIDES, MITICIDES BASF AKTIENGESELLSCHAFT (DE) 1990-05-29 US disclosed
US-4898859-A 2-Oxa-isocephem compounds and compositions containing same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1990-02-06 US disclosed
EP-0351589-A2 3(2H)-Pyridazinone derivatives for controlling snails BASF Aktiengesellschaft (DE) 1990-01-24 EP disclosed
US-4857513-A Diphosphonic acid compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISIWA PHARMACEUTICAL CO., LTD. (JP) 1989-08-15 US disclosed
EP-0320733-A2 2-tert.-butyl-5-isoxazolyl methylthio-3(2H)-pyridazin-3-one derivatives BASF Aktiengesellschaft (DE) 1989-06-21 EP disclosed
CN-88102161-A 2-oxa-isocephem compounds, compositions containing them and processes for their preparation 1988-10-05 CN disclosed
EP-0283970-A2 New peptide compounds, a process for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1988-09-28 EP disclosed
EP-0282895-A2 2-oxa-isocephem compounds, compositions containing same and processes for preparing same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1988-09-21 EP disclosed
EP-0243173-A2 New diphosphonic acid compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1987-10-28 EP disclosed
US-4488897-A Dichloromethyl oxadiazole herbicide antidotes STAUFFER CHEMICAL COMPANY (US) 1984-12-18 US disclosed
US-4488897-A Dichloromethyl oxadiazole herbicide antidotes STAUFFER CHEMICAL COMPANY (US) 1984-12-18 US disclosed
US-RE29577-E Anthraquinone dyestuffs BAYER AKTIENGESELLSCHAFT (DT) 1978-03-14 US disclosed
US-3963763-A Anthraquinone dyestuffs BAYER AKTIENGESELLSCHAFT (DT) 1976-06-15 US disclosed
US-3963763-A Anthraquinone dyestuffs BAYER AKTIENGESELLSCHAFT (DT) 1976-06-15 US disclosed