SCHEMBL5331479

SCHEMBL5331479

O=C(Cl)CCc1nc(-c2ccccc2)no1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.69
TSHR P16473 1/20 0.63
CYP1A2 P05177 2/20 0.62
CYP2C19 P33261 2/20 0.62
CYP2D6 P10635 1/20 0.62
CYP2C9 P11712 1/20 0.62
GAA P10253 1/20 0.61
NPC1 O15118 1/20 0.60
RAB9A P51151 1/20 0.60
L3MBTL1 Q9Y468 1/20 0.60
HDAC1 Q13547 2/20 0.60
HDAC2 Q92769 2/20 0.60
HDAC8 Q9BY41 2/20 0.60
NOTUM Q6P988 1/20 0.59
HPGD P15428 5/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
USP2 O75604 2/20 0.57
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57
LMNA P02545 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5330405 0.88 ALDH1A1 (0.83) ALDH1A1TSHRCYP1A2CYP2C19CYP2D6
SCHEMBL7977105 0.85 ALDH1A1 (0.69) ALDH1A1TSHRCYP1A2CYP2C19CYP2D6
SCHEMBL7977108 0.85 ALDH1A1 (0.69) ALDH1A1TSHRCYP1A2CYP2C19CYP2D6
SCHEMBL11983369 0.85 ALDH1A1 (0.69) ALDH1A1TSHRCYP1A2CYP2C19CYP2D6
SCHEMBL562989 0.82 ALDH1A1 (1.00) ALDH1A1TSHRCYP1A2CYP2C19CYP2D6
SCHEMBL4564362 0.81 HPGD (0.68) ALDH1A1TSHRCYP1A2CYP2C19CYP2D6
SCHEMBL13130280 0.81 TSHR (0.58) ALDH1A1TSHRCYP1A2CYP2C19CYP2D6
SCHEMBL15504863 0.79 RAB9A (0.70) ALDH1A1TSHRCYP1A2CYP2C19CYP2D6
SCHEMBL5717662 0.78 TSHR (1.00) ALDH1A1TSHRNPC1RAB9AHDAC1
SCHEMBL14833395 0.78 CYP1A2 (0.68) ALDH1A1TSHRCYP1A2CYP2C19CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007015744-A1 DISUBSTITUTED THIENYL COMPOUNDS AND THEIR USE AS PHARMACEUTICALS INCYTE CORPORATION (US) 2007-02-08 WO disclosed