SCHEMBL5331629

SCHEMBL5331629

C=Cc1c(C(N)=O)nc(O)c2c1ccn2Cc1ccc(F)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 1/20 0.38
ALDH1A1 P00352 1/20 0.36
GRM2 Q14416 3/20 0.36
MAOB P27338 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
GAA P10253 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC2 Q92769 2/20 0.34
CNR2 P34972 2/20 0.34
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34
FGFR1 P11362 3/20 0.33
FGFR4 P22455 3/20 0.33
DRD2 P14416 1/20 0.33
HTR6 P50406 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6513737 0.85 GAA (0.35) EGLN1ALDH1A1GRM2MAOBCA12
SCHEMBL4801027 0.69 HDAC1 (0.45) EGLN1ALDH1A1MAOBHDAC1HDAC2
SCHEMBL4962821 0.68 L3MBTL1 (0.39) EGLN1GRM2CA12CA1CA2
SCHEMBL4803894 0.67 PDE4B (0.41) ALDH1A1MAOBGAAL3MBTL1MEN1
SCHEMBL3808749 0.64 EGLN1 (0.45) EGLN1MAOB
SCHEMBL5307524 0.64 EGLN1 (0.43) EGLN1GRM2MAOBHDAC1HDAC2
SCHEMBL2145385 0.63 PKM (0.43) ALDH1A1GRM2MAOBGAAMEN1
SCHEMBL18050897 0.63 PKM (0.49) GRM2MAOBGAAMEN1POLB
SCHEMBL4961233 0.63 KDM4E (0.63) ALDH1A1CA12CA1CA2CA9
SCHEMBL2885242 0.62 EGLN1 (0.43) EGLN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756103-A2 PYRROLOPYRIDINE DERIVATIVES AND THEIR USE AS HIV-INTEGRASE INHIBITORS Pfizer, Inc. (US) 2007-02-28 EP disclosed
WO-2005103003-A2 PYRROLOPYRIDINE DERIVATIVES AND THEIR USE AS HIV-INTEGRASE INHIBITORS PFIZER INC. (US) 2005-11-03 WO disclosed