SCHEMBL5332535

SCHEMBL5332535

Cc1ccc2c(c1)CCCN2C(=O)SCC(=O)Nc1cnccc1C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
NPSR1 Q6W5P4 1/20 0.48
KDM4E B2RXH2 2/20 0.46
HTR2C P28335 5/20 0.42
HTR2A P28223 3/20 0.42
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
TSHR P16473 2/20 0.40
HTR2B P41595 4/20 0.40
CYP11B2 P19099 1/20 0.40
POLB P06746 1/20 0.39
MAPT P10636 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
GAA P10253 2/20 0.39
TP53 P04637 1/20 0.39
ALOX15 P16050 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5325413 0.82 ALDH1A1 (0.58) ALDH1A1NPSR1KDM4EHTR2CHTR2A
SCHEMBL5329629 0.80 KDM4E (0.45) ALDH1A1NPSR1KDM4EMEN1KMT2A
SCHEMBL5333492 0.77 HTR2B (0.51) ALDH1A1NPSR1KDM4EHTR2CMEN1
SCHEMBL5328078 0.77 KDM4E (0.51) ALDH1A1NPSR1KDM4EHTR2CHTR2A
SCHEMBL5362566 0.76 KDM4E (0.50) ALDH1A1NPSR1KDM4EMEN1KMT2A
SCHEMBL5370061 0.75 ALDH1A1 (0.46) ALDH1A1NPSR1KDM4EHTR2CHTR2A
SCHEMBL5331465 0.73 KDM4E (0.52) ALDH1A1NPSR1KDM4EMEN1KMT2A
SCHEMBL5324855 0.73 KDM4E (0.48) ALDH1A1NPSR1KDM4EMEN1KMT2A
SCHEMBL5332944 0.72 ALDH1A1 (0.54) ALDH1A1NPSR1KDM4EHTR2CHTR2A
SCHEMBL14346341 0.72 CA1 (0.48) ALDH1A1KDM4EMAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007146230-A2 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS MERCK & CO., INC. (US) 2007-12-21 WO claimed