SCHEMBL5332687

SCHEMBL5332687

COc1ccc2c(c1)c(SCCN(C)C)c(C)n2S(=O)(=O)c1ccc(F)cc1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 18/20 0.56
PTGDR2 Q9Y5Y4 2/20 0.51
PTGDR Q13258 1/20 0.51
HTR1A P08908 1/20 0.43
DRD2 P14416 1/20 0.43
HTR1D P28221 1/20 0.43
HTR1B P28222 1/20 0.43
HTR1E P28566 1/20 0.43
HTR1F P30939 1/20 0.43
HTR7 P34969 1/20 0.43
DRD3 P35462 1/20 0.43
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5425733 0.94 PTGDR2 (0.58) HTR6PTGDR2PTGDR
SCHEMBL5332899 0.94 HTR6 (0.60) HTR6PTGDR2PTGDRHTR1ADRD2
SCHEMBL5332004 0.92 HTR6 (0.58) HTR6PTGDR2PTGDRHTR1ADRD2
SCHEMBL5331612 0.90 HTR6 (0.56) HTR6PTGDR2PTGDRHTR1ADRD2
SCHEMBL5407869 0.90 PTGDR2 (0.54) HTR6PTGDR2PTGDR
SCHEMBL5327800 0.89 HTR6 (0.55) HTR6HTR1ADRD2HTR1DHTR1B
SCHEMBL5330693 0.87 HTR6 (0.53) HTR6PTGDR2PTGDRHTR1ADRD2
SCHEMBL5327989 0.86 HTR6 (0.52) HTR6PTGDR2PTGDRHTR1ADRD2
SCHEMBL5420518 0.86 PTGDR2 (0.45) HTR6PTGDR2PTGDRCYP3A4CYP2D6
SCHEMBL5328966 0.86 PTGDR2 (0.55) HTR6PTGDR2PTGDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007020653-A1 THIOETHER DERIVATIVES AS FUNCTIONAL 5-HT6 LIGANDS SUVEN LIFE SCIENCES LIMITED (IN) 2007-02-22 WO disclosed