SCHEMBL5333399

SCHEMBL5333399

CCCc1nn(C)c2c(Nc3ccc(F)cc3)nc(-c3ccc(F)cc3)nc12

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 5/20 0.41
ABCG2 Q9UNQ0 1/20 0.40
KDM1A O60341 2/20 0.39
PDE4B Q07343 3/20 0.38
PDE4D Q08499 3/20 0.38
HTR2C P28335 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
RXRA P19793 1/20 0.37
NR4A2 P43354 1/20 0.37
NPC1 O15118 1/20 0.37
HTT P42858 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MEN1 O00255 2/20 0.36
HPGD P15428 2/20 0.36
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 1/20 0.36
USP2 O75604 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5372075 0.99 PDE5A (0.40) PDE5AABCG2KDM1APDE4BPDE4D
Hydrochloric Acid SCHEMBL5360340 0.89 CHRNA7 (0.48)
Hydrochloric Acid SCHEMBL5357538 0.88 PDE5A (0.39) PDE5AABCG2PDE4BPDE4DHDAC1
SCHEMBL5365432 0.87 ABCG2 (0.50) PDE5AABCG2PDE4BPDE4DHDAC1
Hydrochloric Acid SCHEMBL5328212 0.87 ABCG2 (0.45) PDE5AABCG2HDAC1HDAC6SMN1; SMN2
Hydrochloric Acid SCHEMBL5328910 0.86 PDE5A (0.38) PDE5AABCG2HDAC1HDAC6NPC1
Hydrochloric Acid SCHEMBL5358447 0.86 ABCG2 (0.49) PDE5AABCG2PDE4BPDE4DHDAC1
SCHEMBL2857503 0.86 PDE5A (0.38) PDE5AHTR2CHDAC1HDAC6NPC1
Hydrochloric Acid SCHEMBL6103394 0.86 ABCG2 (0.48) PDE5AABCG2PDE4BPDE4DHDAC1
Hydrochloric Acid SCHEMBL5369756 0.86 KMT2A (0.41) HTTMEN1HPGDKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1814885-A2 NOVEL BICYCLIC HETEROCYCLIC COMPOUNDS, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM Reddy US Therapeutics, Inc. (US) 2007-08-08 EP disclosed
WO-2006073610-A2 NOVEL BICYCLIC HETEROCYCLIC COMPOUNDS, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM REDDY US THERAPEUTICS, INC. (US) 2006-07-13 WO disclosed