SCHEMBL5333874

SCHEMBL5333874

O=C(NNC(=S)Nc1ccccc1)c1ccc2c(c1)OCO2

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.77
RAB9A P51151 8/20 0.77
SMN1; SMN2 Q16637 7/20 0.77
MAPT P10636 4/20 0.77
ALDH1A1 P00352 4/20 0.77
PKM P14618 2/20 0.73
GAA P10253 6/20 0.68
KMT2A Q03164 2/20 0.68
LMNA P02545 2/20 0.68
MEN1 O00255 1/20 0.68
P2RX2 Q9UBL9 2/20 0.66
P2RX4 Q99571 2/20 0.66
P2RX5 Q93086 1/20 0.66
P2RX7 Q99572 1/20 0.66
CYP1A2 P05177 2/20 0.63
CYP2D6 P10635 2/20 0.63
EGFR P00533 1/20 0.62
NFKB1 P19838 2/20 0.61
NFKB2 Q00653 2/20 0.61
RELA Q04206 2/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11238457 0.85 RAB9A (1.00) NPC1RAB9ASMN1; SMN2MAPTALDH1A1
SCHEMBL4409690 0.78 RAB9A (0.64) NPC1RAB9ASMN1; SMN2MAPTALDH1A1
SCHEMBL13547676 0.77 GAA (1.00) NPC1RAB9ASMN1; SMN2MAPTALDH1A1
SCHEMBL19478515 0.76 GAA (1.00) NPC1RAB9ASMN1; SMN2MAPTALDH1A1
SCHEMBL4727186 0.75 RAB9A (0.81) NPC1RAB9ASMN1; SMN2MAPTALDH1A1
SCHEMBL5330501 0.75 NPC1 (1.00) NPC1RAB9ASMN1; SMN2MAPTALDH1A1
SCHEMBL12098605 0.75 MAPT (0.72) NPC1RAB9ASMN1; SMN2MAPTALDH1A1
SCHEMBL3519624 0.75 RAB9A (0.70) NPC1RAB9ASMN1; SMN2MAPTALDH1A1
SCHEMBL12827566 0.74 RAB9A (0.78) NPC1RAB9ASMN1; SMN2MAPTALDH1A1
SCHEMBL12083878 0.74 RAB9A (0.58) NPC1RAB9ASMN1; SMN2MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007047394-A2 THIOTRIAZOLYL DERIVATIVES EPIX DELAWARE, INC. (US) 2007-04-26 WO disclosed